SCHEMBL11196264

SCHEMBL11196264

NCCNC(=O)COc1ccc(CC(N)=O)cc1

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.49
PTPN1 P18031 1/20 0.49
HDAC1 Q13547 1/20 0.49
LMNA P02545 1/20 0.47
PKM P14618 1/20 0.47
PPARD Q03181 1/20 0.47
ALDH1A1 P00352 1/20 0.47
RAB9A P51151 1/20 0.46
MEN1 O00255 1/20 0.46
PPARG P37231 1/20 0.46
HTT P42858 1/20 0.46
KMT2A Q03164 1/20 0.46
NCOA2 Q15596 1/20 0.46
NCOA1 Q15788 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
NR2E3 Q9Y5X4 1/20 0.46
NCOR2 Q9Y618 1/20 0.46
NCOA3 Q9Y6Q9 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22257276 0.80 KMT2A (0.58) KDM4EHDAC1ALDH1A1MEN1HTT
SCHEMBL7890148 0.80 NPC1 (0.63) KDM4EPTPN1ALDH1A1RAB9AMEN1
Hydrochloric Acid SCHEMBL20529584 0.79 KMT2A (0.56) KDM4EHDAC1ALDH1A1MEN1HTT
Hydrochloric Acid SCHEMBL11571294 0.78 NPC1 (0.61) KDM4EPTPN1ALDH1A1RAB9AMEN1
SCHEMBL23582957 0.76 ALOX15 (0.57) ALDH1A1MEN1KMT2A
SCHEMBL8475224 0.76 TBXAS1 (0.55) LMNA
SCHEMBL7601684 0.76 CA2 (0.55) KDM4ELMNA
SCHEMBL1048553 0.75 SMN1; SMN2 (0.70) KDM4EPTPN1LMNAALDH1A1RAB9A
SCHEMBL11191751 0.75 HTT (0.65) LMNAPKMALDH1A1RAB9AMEN1
SCHEMBL23599248 0.75 TDP1 (0.52) KDM4ELMNANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4387099-A Alkanolamine derivatives IMPERIAL CHEMICAL INDUSTRIES LIMITED (GB) 1983-06-07 US disclosed
US-4327113-A DRUGS FOR TREATMENT OF HEART DISEASES, ADRENERGIC BLOCKING AGENTS, ETC IMPERIAL CHEMICAL INDUSTRIES LIMITED (GB) 1982-04-27 US disclosed
US-4260632-A ADRENERGIC BLOCKING AGENTS, CARDIOVASCULAR DISORDERS IMPERIAL CHEMICAL INDUSTRIES LIMITED (GB) 1981-04-07 US disclosed
US-4221807-A ADRENERGIC BLOCKING AGENTS IMPERIAL CHEMICAL INDUSTRIES LIMITED (GB) 1980-09-09 US disclosed
US-4141987-A HYPOTENSIVE, ADRENERGIC BLOCKING AGENT IMPERIAL CHEMICAL INDUSTRIES LIMITED (GB) 1979-02-27 US disclosed