Bromide

Bromide

SCHEMBL11199816

Br.O=C1CCc2cc(N3CCNCC3)ccc2N1

nearest known ligand 0.52

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 known ✓ P31645 4/20 0.51
ADRB1 known ✓ P08588 3/20 0.44
HTR1A known ✓ P08908 2/20 0.43
SLC6A2 known ✓ P23975 2/20 0.43
SLC6A3 known ✓ Q01959 2/20 0.43
HTR3A known ✓ P46098 2/20 0.43
SIGMAR1 known ✓ Q99720 2/20 0.43
CRBN Q96SW2 5/20 0.52
PDE3B Q13370 2/20 0.52
PDE3A Q14432 2/20 0.52
TBXAS1 P24557 1/20 0.52
KCNH2 Q12809 2/20 0.51
NR3C1 P04150 1/20 0.51
PGR P06401 1/20 0.51
DDB1 Q16531 2/20 0.47
MAPKAPK2 P49137 2/20 0.46
NPC1 O15118 1/20 0.44
MAPK13 O15264 1/20 0.44
MAPK12 P53778 1/20 0.44
MAPK11 Q15759 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7274510 0.98 CRBN (0.53) CRBNPDE3BPDE3ATBXAS1SLC6A4
Bromide SCHEMBL11198697 0.88 CRBN (0.52) CRBNSLC6A4DDB1ADRB1NPC1
Bromide SCHEMBL9825246 0.87 MAPKAPK2 (0.52) MAPKAPK2ADRB1
SCHEMBL9824743 0.85 MAPKAPK2 (0.53) MAPKAPK2ADRB1
SCHEMBL8880352 0.83 CRBN (0.53) CRBNPDE3BPDE3ATBXAS1SLC6A4
SCHEMBL11196268 0.82 CRBN (0.52) CRBNPDE3BPDE3ATBXAS1SLC6A4
SCHEMBL8807339 0.80 SLC6A4 (0.52) CRBNPDE3BPDE3ATBXAS1SLC6A4
Hydrochloric Acid SCHEMBL7286588 0.79 SMYD3 (0.50) CRBNPDE3BPDE3ATBXAS1SLC6A4
SCHEMBL11197711 0.78 PDE3B (0.53) CRBNPDE3BPDE3ATBXAS1SLC6A4
SCHEMBL11194801 0.78 SLC6A4 (0.64) CRBNPDE3BPDE3ATBXAS1SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4415572-A CARDIOTONIC AND INOTROPIC AGENTS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1983-11-15 US disclosed