SCHEMBL11200295

SCHEMBL11200295

O=C(Nc1nccs1)c1c(C(F)(F)F)nc2ccccc2c1O

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.54
LMNA P02545 7/20 0.53
MAPT P10636 3/20 0.53
HPGD P15428 2/20 0.53
NPC1 O15118 4/20 0.51
RAB9A P51151 4/20 0.51
MEN1 O00255 5/20 0.50
KMT2A Q03164 5/20 0.50
HTT P42858 2/20 0.50
CYP1A2 P05177 2/20 0.48
L3MBTL1 Q9Y468 4/20 0.48
KDM4E B2RXH2 3/20 0.48
POLB P06746 2/20 0.48
MCL1 Q07820 1/20 0.48
CTDSP1 Q9GZU7 1/20 0.48
SAE1 Q9UBE0 1/20 0.48
UBA2 Q9UBT2 1/20 0.48
SCD O00767 1/20 0.47
SMN1; SMN2 Q16637 3/20 0.47
METAP2 P50579 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11148451 0.86 NPC1 (0.45) ALDH1A1LMNAMAPTHPGDNPC1
SCHEMBL11200589 0.86 NPC1 (0.43) ALDH1A1LMNAMAPTHPGDNPC1
SCHEMBL11148448 0.84 HTT (0.46) LMNAMAPTHPGDNPC1RAB9A
SCHEMBL11208407 0.83 ALDH1A1 (0.45) ALDH1A1LMNAMAPTHPGDNPC1
SCHEMBL11192028 0.83 HPGDS (0.52) ALDH1A1LMNAMAPTNPC1RAB9A
SCHEMBL9775626 0.83 RAB9A (0.49) ALDH1A1LMNAMAPTHPGDNPC1
SCHEMBL9775616 0.82 RAB9A (0.50) LMNAMAPTHPGDNPC1RAB9A
SCHEMBL9775604 0.81 RAB9A (0.49) ALDH1A1LMNAMAPTHPGDNPC1
SCHEMBL11200852 0.81 NPC1 (0.51) ALDH1A1LMNAMAPTNPC1RAB9A
SCHEMBL9775653 0.79 MEN1 (0.46) ALDH1A1LMNAMAPTHPGDNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4299831-A 2-Trifluoromethyl-3-quinoline carboxamides, analgesic and anti-inflammatory compositions and methods employing them ROUSSEL UCLAF (FR) 1981-11-10 US claimed
EP-0012639-B1 QUINOLEIN-3-CARBOXYLIC ACID DERIVATIVES, PROCESS FOR THEIR PREPARATION, THEIR USE IN MEDICINES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM ROUSSEL-UCLAF (FR) 1983-09-07 EP disclosed
US-4299831-A 2-Trifluoromethyl-3-quinoline carboxamides, analgesic and anti-inflammatory compositions and methods employing them ROUSSEL UCLAF (FR) 1981-11-10 US disclosed
EP-0012639-A2 Quinolein-3-carboxylic acid derivatives, process for their preparation, their use in medicines and pharmaceutical compositions containing them ROUSSEL-UCLAF (FR) 1980-06-25 EP disclosed