SCHEMBL11200643

SCHEMBL11200643

C=Cn1cc(C(=O)O)c(=O)c2cc(F)c(N3CCN(C(=O)OCC)CC3)nc21

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.55
CYP2C9 P11712 1/20 0.55
ATP6V1B2 P21281 1/20 0.55
TBXA2R P21731 1/20 0.55
EDNRA P25101 1/20 0.55
TARBP2 Q15633 1/20 0.55
ALDH1A1 P00352 3/20 0.43
KDM4E B2RXH2 2/20 0.43
HSD17B10 Q99714 3/20 0.42
KMT2A Q03164 5/20 0.42
DPP4 P27487 2/20 0.41
CHRM2 P08172 1/20 0.41
DRD1 P21728 1/20 0.41
MAPT P10636 3/20 0.41
MEN1 O00255 3/20 0.41
MAPK1 P28482 1/20 0.41
CASP1 P29466 1/20 0.41
CASP7 P55210 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41
HTT P42858 4/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11035359 0.87 LMNA (0.72) LMNACYP2C9ATP6V1B2TBXA2REDNRA
SCHEMBL9437305 0.84 DPP4 (0.58) LMNACYP2C9ATP6V1B2TBXA2REDNRA
SCHEMBL11277560 0.81 LMNA (0.59) LMNACYP2C9ATP6V1B2TBXA2REDNRA
SCHEMBL10521403 0.81 LMNA (0.70) LMNACYP2C9ATP6V1B2TBXA2REDNRA
SCHEMBL11092618 0.79 LMNA (0.61) LMNACYP2C9ATP6V1B2TBXA2REDNRA
SCHEMBL11089508 0.78 KDM4E (0.51) LMNACYP2C9ATP6V1B2TBXA2REDNRA
SCHEMBL18213620 0.78 LMNA (0.65) LMNACYP2C9ATP6V1B2TBXA2REDNRA
SCHEMBL11714386 0.77 SMN1; SMN2 (0.44) LMNACYP2C9ALDH1A1KDM4EHSD17B10
SCHEMBL11269349 0.77 LMNA (0.52) LMNACYP2C9ATP6V1B2TBXA2REDNRA
SCHEMBL9437310 0.77 DPP4 (0.50) LMNACYP2C9ATP6V1B2TBXA2REDNRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4382937-A Naphthyridine derivatives and their use as anti-bacterials DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 1983-05-10 US disclosed
US-4359578-A Naphthyridine derivatives and salts thereof useful as antibacterial agents DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 1982-11-16 US disclosed
US-4352803-A BACTERICIDES DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 1982-10-05 US disclosed
EP-0009425-B1 NOVEL NAPHTYRIDINE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Société anonyme dite: LABORATOIRE ROGER BELLON (FR) 1982-01-27 EP disclosed
EP-0009425-A1 Novel naphtyridine derivatives and pharmaceutical compositions containing them Société anonyme dite: LABORATOIRE ROGER BELLON (FR) 1980-04-02 EP disclosed