SCHEMBL11200904

SCHEMBL11200904

CSc1ncc(-c2ccc(C)nc2)c(=O)n1C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.39
KDM4E B2RXH2 2/20 0.37
LMNA P02545 1/20 0.37
MEN1 O00255 1/20 0.37
NPC1 O15118 1/20 0.37
CRHBP P24387 1/20 0.37
RAB9A P51151 1/20 0.37
KMT2A Q03164 1/20 0.37
CRHR2 Q13324 1/20 0.37
PTGS2 P35354 2/20 0.36
SLC22A12 Q96S37 1/20 0.36
HPGD P15428 2/20 0.35
POLB P06746 1/20 0.35
DAO P14920 1/20 0.35
PDE3B Q13370 3/20 0.35
PDE3A Q14432 3/20 0.35
MAPK1 P28482 1/20 0.35
CASP1 P29466 1/20 0.35
HSD17B10 Q99714 1/20 0.35
SYK P43405 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2861659 0.77 ALDH1A1 (0.39) ALDH1A1KDM4ELMNAHPGDDAO
SCHEMBL2070913 0.72 CRHR1 (0.37) KDM4ELMNAMEN1RAB9AKMT2A
SCHEMBL27250753 0.71 CYP1A2 (0.41) ALDH1A1KDM4EPTGS2SLC22A12HPGD
SCHEMBL2070835 0.69 RXFP1 (0.37) ALDH1A1KDM4ELMNAMEN1NPC1
SCHEMBL11491285 0.67 RXFP1 (0.36) ALDH1A1KDM4ELMNAMEN1NPC1
SCHEMBL15026014 0.64 HPGDS (0.44) ALDH1A1MEN1NPC1RAB9AKMT2A
SCHEMBL676678 0.64 HPGDS (0.56) NPC1RAB9APTGS2PIK3CAHPGDS
SCHEMBL11203629 0.64 KLKB1 (0.42) ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL22932832 0.64 KDM4E (0.51) ALDH1A1KDM4ELMNAMEN1NPC1
SCHEMBL10986060 0.64 ALDH1A1 (0.54) ALDH1A1KDM4ELMNAMEN1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0083186-A2 Thiazole derivatives as H2-receptor antagonists ELI LILLY AND COMPANY (US) 1983-07-06 EP disclosed