SCHEMBL11201034

SCHEMBL11201034

COc1ccc(C(=O)N2CCN(c3ccc4c(c3)NC(=O)CC4)CC2)cc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 1/20 0.66
PGR P06401 1/20 0.66
SLC6A4 P31645 1/20 0.66
KCNH2 Q12809 1/20 0.66
PDE3B Q13370 1/20 0.66
PDE3A Q14432 1/20 0.66
ALDH1A1 P00352 7/20 0.57
HTT P42858 2/20 0.57
KDM4E B2RXH2 1/20 0.57
DRD2 P14416 2/20 0.57
DRD4 P21917 1/20 0.57
DRD3 P35462 1/20 0.57
GAA P10253 1/20 0.55
MAPT P10636 5/20 0.53
LMNA P02545 4/20 0.53
MEN1 O00255 3/20 0.53
KMT2A Q03164 3/20 0.53
TSHR P16473 1/20 0.52
SMN1; SMN2 Q16637 4/20 0.51
GLA P06280 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11202820 0.92 NR3C1 (0.78) NR3C1PGRSLC6A4KCNH2PDE3B
Water SCHEMBL11200345 0.91 NR3C1 (0.76) NR3C1PGRSLC6A4KCNH2PDE3B
Water SCHEMBL11200349 0.91 NR3C1 (0.76) NR3C1PGRSLC6A4KCNH2PDE3B
SCHEMBL8495619 0.88 PDE3B (0.85) NR3C1PGRSLC6A4KCNH2PDE3B
SCHEMBL11192867 0.86 KCNH2 (0.58) NR3C1PGRSLC6A4KCNH2PDE3B
SCHEMBL11202917 0.85 PDE3B (0.57) NR3C1PGRSLC6A4KCNH2PDE3B
SCHEMBL8499623 0.85 PDE3B (0.69) NR3C1PGRSLC6A4KCNH2PDE3B
SCHEMBL11042441 0.83 NR3C1 (0.66) NR3C1PGRSLC6A4KCNH2PDE3B
SCHEMBL11200540 0.82 NR3C1 (0.54) NR3C1PGRSLC6A4KCNH2PDE3B
SCHEMBL11196576 0.81 KCNH2 (0.69) NR3C1PGRSLC6A4KCNH2PDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4415572-A CARDIOTONIC AND INOTROPIC AGENTS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1983-11-15 US disclosed