SCHEMBL11204329

SCHEMBL11204329

CC(CNC(=O)Cc1ccccc1)NCC(O)COc1cccc2c1OCCO2

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 8/20 0.46
ADRB1 P08588 7/20 0.46
MTNR1A P48039 4/20 0.46
ADRB3 P13945 1/20 0.42
MEN1 O00255 1/20 0.41
ALDH1A1 P00352 1/20 0.41
KMT2A Q03164 1/20 0.41
ABCB1 P08183 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11201763 0.84 MTNR1A (0.45) ADRB2ADRB1MTNR1AMEN1KMT2A
SCHEMBL11476015 0.82 MTNR1A (0.49) ADRB2ADRB1MTNR1AADRB3ALDH1A1
SCHEMBL11570223 0.79 MEN1 (0.64) ADRB2ADRB1ADRB3MEN1ALDH1A1
SCHEMBL11476025 0.77 MTNR1A (0.48) ADRB2ADRB1MTNR1AADRB3MEN1
SCHEMBL7518458 0.77 MTNR1A (0.69) MTNR1AALDH1A1
SCHEMBL11478876 0.77 MTNR1A (0.48) ADRB2ADRB1MTNR1AADRB3ALDH1A1
SCHEMBL11478895 0.74 MTNR1A (0.50) ADRB2ADRB1MTNR1AADRB3ABCB1
SCHEMBL11266560 0.70 TACR1 (0.39) MTNR1AALDH1A1
SCHEMBL13533389 0.68 MTNR1A (0.53) MTNR1A
SCHEMBL11652084 0.68 ADRB3 (0.54) ADRB2ADRB1ADRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4387099-A Alkanolamine derivatives IMPERIAL CHEMICAL INDUSTRIES LIMITED (GB) 1983-06-07 US disclosed
US-4327113-A DRUGS FOR TREATMENT OF HEART DISEASES, ADRENERGIC BLOCKING AGENTS, ETC IMPERIAL CHEMICAL INDUSTRIES LIMITED (GB) 1982-04-27 US disclosed
US-4260632-A ADRENERGIC BLOCKING AGENTS, CARDIOVASCULAR DISORDERS IMPERIAL CHEMICAL INDUSTRIES LIMITED (GB) 1981-04-07 US disclosed
US-4221807-A ADRENERGIC BLOCKING AGENTS IMPERIAL CHEMICAL INDUSTRIES LIMITED (GB) 1980-09-09 US disclosed
US-4141987-A HYPOTENSIVE, ADRENERGIC BLOCKING AGENT IMPERIAL CHEMICAL INDUSTRIES LIMITED (GB) 1979-02-27 US disclosed