SCHEMBL11208313

SCHEMBL11208313

CNc1nc(N2CCNCC2)nc2sc(C(C)C)cc12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 3/20 0.42
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 2/20 0.41
HTR2C P28335 1/20 0.39
KHK P50053 1/20 0.38
CASP1 P29466 1/20 0.38
CASP4 P49662 1/20 0.38
CASP5 P51878 1/20 0.38
PLK4 O00444 1/20 0.37
PAK4 O96013 1/20 0.37
HTR3A P46098 2/20 0.36
HRH4 Q9H3N8 2/20 0.36
TSHR P16473 1/20 0.36
HRH1 P35367 1/20 0.36
PRKCI P41743 2/20 0.35
USP2 O75604 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
APAF1 O14727 1/20 0.34
POLB P06746 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11202691 0.84 KHK (0.42) HTR2AKDM4EALDH1A1HTR2CKHK
Hydrochloric Acid SCHEMBL11201994 0.82 KHK (0.41) HTR2AKDM4EALDH1A1HTR2CKHK
SCHEMBL11200730 0.82 KDM4E (0.49) HTR2AKDM4EALDH1A1HTR2CCASP1
SCHEMBL11199721 0.81 P2RY12 (0.50) HTR2AKDM4EALDH1A1HTR2CKHK
SCHEMBL11204604 0.79 P2RY12 (0.42) HTR2AKDM4EALDH1A1HTR2CKHK
SCHEMBL11200417 0.77 MEN1 (0.45) KDM4EALDH1A1TSHRSMN1; SMN2MAPT
SCHEMBL11201826 0.77 CETP (0.42) HTR2AKDM4EALDH1A1HTR2CKHK
SCHEMBL11205604 0.74 HTR2C (0.65) HTR2AKDM4EALDH1A1HTR2CKHK
SCHEMBL11200202 0.74 KHK (0.38) HTR2AKDM4EALDH1A1HTR2CKHK
SCHEMBL11206366 0.73 HTR2A (0.39) HTR2AKDM4EALDH1A1HTR2CKHK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0082023-A2 Thienopyrimidine derivatives, their preparation and their medical use SANKYO COMPANY LIMITED (JP) 1983-06-22 EP disclosed