SCHEMBL11209050

SCHEMBL11209050

CCC(=O)Nc1ccc(O)c(C#N)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.51
ALDH1A1 P00352 4/20 0.49
RAB9A P51151 3/20 0.49
KDM4E B2RXH2 1/20 0.49
HPGD P15428 1/20 0.49
TSHR P16473 1/20 0.48
POLB P06746 3/20 0.47
NR4A1 P22736 1/20 0.47
PGR P06401 1/20 0.47
GAA P10253 3/20 0.47
MAPT P10636 2/20 0.47
CYP1A2 P05177 2/20 0.47
CYP2C19 P33261 2/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
NPC1 O15118 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C9 P11712 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
CA12 O43570 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24061321 0.83 TSHR (0.61) CYP3A4ALDH1A1RAB9AKDM4EHPGD
SCHEMBL7754593 0.82 ALDH1A1 (0.65) CYP3A4ALDH1A1RAB9AKDM4EHPGD
SCHEMBL17365323 0.80 CYP3A4 (0.61) CYP3A4ALDH1A1RAB9AKDM4EHPGD
SCHEMBL11297032 0.78 KMT2A (0.49) ALDH1A1RAB9AKDM4EHPGDPGR
SCHEMBL20852437 0.77 AR (0.62)
SCHEMBL14241325 0.76 TSHR (0.64) CYP3A4ALDH1A1RAB9AKDM4EHPGD
SCHEMBL9645123 0.76 CYP3A4 (0.56) CYP3A4ALDH1A1RAB9AKDM4EHPGD
SCHEMBL10816910 0.76 MEN1 (0.56) ALDH1A1RAB9AHPGDTSHRPOLB
SCHEMBL10815837 0.76 KMT2A (0.56) ALDH1A1RAB9AHPGDTSHRPOLB
SCHEMBL14266363 0.75 SAE1 (0.57) ALDH1A1RAB9AKDM4EHPGDTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0035734-B1 1-(ACYLAMINO-ARYLOXY-)2-HYDROXY-3-ALKINYL-AMINO PROPANES AND PROCESSES FOR THEIR MANUFACTURE C.H. BOEHRINGER SOHN (DE) 1983-09-21 EP disclosed
US-4344964-A HYPOTENSIVE AGENTS, ANTIARRHYTHMIA AGENTS C. H. BOEHRINGER SOHN (DE) 1982-08-17 US disclosed
EP-0035734-A1 1-(Acylamino-aryloxy-)2-hydroxy-3-alkinyl-amino propanes and processes for their manufacture C.H. BOEHRINGER SOHN (DE) 1981-09-16 EP disclosed