SCHEMBL11209428

SCHEMBL11209428

CSC(C)(C#N)c1cccc(C(=O)c2ccccc2)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
SRD5A2 P31213 1/20 0.46
VNN1 O95497 4/20 0.44
ABCC9 O60706 1/20 0.42
ABCC8 Q09428 1/20 0.42
KCNJ11 Q14654 1/20 0.42
KCNJ8 Q15842 1/20 0.42
PBRM1 Q86U86 1/20 0.41
MAPT P10636 2/20 0.40
PTGS1 P23219 2/20 0.40
CXCR1 P25024 2/20 0.40
CXCR2 P25025 2/20 0.40
PTGS2 P35354 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
ALDH1A1 P00352 2/20 0.40
RECQL P46063 1/20 0.40
ACHE P22303 1/20 0.40
KDM4E B2RXH2 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28294064 0.82 ATM (0.53) ATMTDP1L3MBTL1SRD5A2VNN1
SCHEMBL11213960 0.82 ATM (0.41) ATMTDP1L3MBTL1SRD5A2VNN1
SCHEMBL11213109 0.81 L3MBTL1 (0.40) ATMTDP1L3MBTL1SRD5A2VNN1
SCHEMBL11480384 0.78 ATM (0.52) ATMTDP1L3MBTL1SRD5A2VNN1
SCHEMBL3684740 0.76 ATM (0.63) ATMTDP1L3MBTL1SRD5A2VNN1
SCHEMBL11210271 0.76 PPARA (0.44) MAPTSMN1; SMN2ALDH1A1RECQLHPGD
SCHEMBL11482204 0.75 ATM (0.45) ATMTDP1L3MBTL1SRD5A2VNN1
SCHEMBL548283 0.75 L3MBTL1 (0.61) ATMTDP1L3MBTL1SRD5A2VNN1
SCHEMBL11210711 0.74 AKR1C3 (0.39) ATMTDP1MAPTPTGS1SMN1; SMN2
SCHEMBL7488968 0.73 ATM (0.59) ATMTDP1L3MBTL1SRD5A2VNN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0025262-B1 ALPHA-THIO-ALPHA-ARYL-SUBSTITUTED ALKANONITRILES, PROCESS FOR THEIR PREPARATION, PROCESS FOR PREPARING ALPHA-ARYL-SUBSTITUTED ALKANONITRILES AND THE CORRESPONDING CARBOXYLIC ACIDS THEREFROM AND PROCESS FOR PREPARING INTERMEDIATES SAGAMI CHEMICAL RESEARCH CENTER (JP) 1983-10-05 EP disclosed
US-4340740-A Alpha-thio-alpha-aryl-substituted alkanonitrile and process for preparing alpha-aryl-substituted alkanonitrile therefrom SAGAMI CHEMICAL RESEARCH CENTER (JP) 1982-07-20 US disclosed
EP-0025262-A2 Alpha-thio-alpha-aryl-substituted alkanonitriles, process for their preparation, process for preparing alpha-aryl-substituted alkanonitriles and the corresponding carboxylic acids therefrom and process for preparing intermediates SAGAMI CHEMICAL RESEARCH CENTER (JP) 1981-03-18 EP disclosed