SCHEMBL11211906

SCHEMBL11211906

CC(=O)NC1CCc2n[nH]cc2C1

nearest known ligand 0.54

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 9/20 0.54
MTNR1B P49286 7/20 0.54
CA1 P00915 4/20 0.37
CA2 P00918 4/20 0.37
CA12 O43570 2/20 0.37
CA7 P43166 2/20 0.37
CA14 Q9ULX7 2/20 0.37
CA9 Q16790 1/20 0.36
ATM Q13315 1/20 0.36
ACHE P22303 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11212845 0.95 MTNR1A (0.49) MTNR1AMTNR1BCA1CA2CA12
SCHEMBL11232532 0.85 MTNR1A (0.57) MTNR1AMTNR1BCA1CA2CA12
SCHEMBL2205376 0.83 EPHX2 (0.47) MTNR1AMTNR1B
SCHEMBL24263104 0.79 MTNR1A (0.50) MTNR1AMTNR1BCA1CA2CA12
SCHEMBL11275699 0.76 MTNR1A (0.66) MTNR1AMTNR1BCA1CA2CA12
SCHEMBL13787618 0.73 TOP2A (0.37) MTNR1AMTNR1B
SCHEMBL16082811 0.72 MTNR1A (0.52) MTNR1AMTNR1BCA1CA2CA12
SCHEMBL5053490 0.72 MTNR1A (0.64) MTNR1AMTNR1BCA1CA2ACHE
SCHEMBL5053493 0.72 MTNR1A (0.64) MTNR1AMTNR1BCA1CA2ACHE
SCHEMBL12432084 0.72 PDK1 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014145512-A2 POTENT SMALL MOLECULE INHIBITORS OF AUTOPHAGY, AND METHODS OF USE THEREOF PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2014-09-18 WO disclosed
EP-0013789-B1 AMINO-SUBSTITUTED 4,5,6,7-TETRAHYDRO-1H (OR 2H)-INDAZOLES, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM ELI LILLY AND COMPANY (US) 1983-02-02 EP disclosed
EP-0013789-A1 Amino-substituted 4,5,6,7-tetrahydro-1H (or 2H)-indazoles, their preparation and pharmaceutical compositions containing them ELI LILLY AND COMPANY (US) 1980-08-06 EP disclosed