SCHEMBL11212751

SCHEMBL11212751

O=C(O)CCC[CH]NC(=O)c1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 3/20 0.49
HDAC1 Q13547 3/20 0.49
HDAC7 Q8WUI4 3/20 0.49
HDAC2 Q92769 3/20 0.49
HDAC8 Q9BY41 3/20 0.49
HDAC6 Q9UBN7 3/20 0.49
HDAC4 P56524 2/20 0.49
HDAC10 Q969S8 2/20 0.49
HDAC11 Q96DB2 2/20 0.49
HDAC9 Q9UKV0 2/20 0.49
HDAC5 Q9UQL6 2/20 0.49
MAPK1 P28482 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
ADRA1A P35348 1/20 0.47
SLC6A3 Q01959 1/20 0.47
TOP1 P11387 1/20 0.46
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
TBXAS1 P24557 4/20 0.46
MAPT P10636 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11634994 0.83 NR1H4 (0.58) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL1556345 0.83 NAAA (0.54) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL1416822 0.81 NAAA (0.57) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL1416655 0.79 RAB9A (0.49) HDAC3HDAC1HDAC7HDAC2HDAC8
SCHEMBL4611015 0.76 NPC1 (0.54) HDAC3HDAC1HDAC7HDAC2HDAC8
SCHEMBL727648 0.76 RAB9A (0.53) HDAC3HDAC1HDAC7HDAC2HDAC8
SCHEMBL692327 0.74 RAB9A (0.49) HDAC3HDAC1HDAC7HDAC2HDAC8
SCHEMBL18151630 0.74 HDAC3 (0.58) HDAC3HDAC1HDAC2HDAC8SMN1; SMN2
Benzoic Acid Hydrazide SCHEMBL11870297 0.74 HDAC3 (0.60) HDAC3HDAC1HDAC7HDAC2HDAC8
Pimelic Acid SCHEMBL28874757 0.74 HDAC1 (0.66) HDAC3HDAC1HDAC7HDAC2HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4311704-A ANTIBIOTICS MERCK & CO., INC. (US) 1982-01-19 US disclosed
EP-0001264-A1 Substituted N-methylene derivatives of thienamycin sulfoxide and sulfone and their preparation MERCK & CO. INC. (US) 1979-04-04 EP disclosed