SCHEMBL11213151

SCHEMBL11213151

O=C1CCC(c2ccsc2)=NN1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.59
PDE3B Q13370 13/20 0.51
PDE3A Q14432 13/20 0.51
PDE4A P27815 7/20 0.48
PDE4B Q07343 7/20 0.48
PDE4C Q08493 7/20 0.48
PDE4D Q08499 7/20 0.48
KCNH2 Q12809 1/20 0.48
LMNA P02545 2/20 0.46
MAPT P10636 2/20 0.46
NPY1R P25929 1/20 0.46
NPY2R P49146 1/20 0.46
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
TSHR P16473 1/20 0.44
MAPK1 P28482 1/20 0.44
CYP2C19 P33261 1/20 0.44
KMT2A Q03164 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6849455 0.84 AXL (0.58) SMN1; SMN2PDE3BPDE3ACYP3A4CYP2C9
SCHEMBL10558463 0.79 PDE3B (0.44) SMN1; SMN2PDE3BPDE3APDE4APDE4B
SCHEMBL10353452 0.79 SMN1; SMN2 (0.81) SMN1; SMN2PDE3BPDE3APDE4APDE4B
SCHEMBL10770050 0.78 PDE3B (0.43) SMN1; SMN2PDE3BPDE3APDE4APDE4B
SCHEMBL10770060 0.78 GPR119 (0.45) SMN1; SMN2PDE3BPDE3APDE4APDE4B
SCHEMBL2592010 0.78 GPR119 (0.72)
SCHEMBL10518299 0.78 GPR119 (0.59) SMN1; SMN2PDE3BPDE3APDE4APDE4B
SCHEMBL7263634 0.77 KCNH2 (0.73) SMN1; SMN2PDE3BPDE3APDE4APDE4B
SCHEMBL9369671 0.76 PDE3B (0.53) SMN1; SMN2PDE3BPDE3APDE4APDE4B
SCHEMBL10473667 0.74 KCNH2 (0.50) SMN1; SMN2PDE3BPDE3APDE4APDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0029103-B1 6- AND 8-HETEROARYL-1,2,4-TRIAZOLO(4,3-B)PYRIDAZINES AMERICAN CYANAMID COMPANY (US) 1983-05-18 EP disclosed
US-4260756-A TRANQUILIZERS AMERICAN CYANAMID COMPANY (US) 1981-04-07 US disclosed