SCHEMBL11214020

SCHEMBL11214020

N#CC(Sc1nc2ccccc2s1)c1cccc(Oc2ccccc2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.40
HPGD P15428 4/20 0.40
ALOX15 P16050 2/20 0.40
HSD17B10 Q99714 2/20 0.40
TDP1 Q9NUW8 2/20 0.40
ADRA2A P08913 1/20 0.40
FBP1 P09467 1/20 0.40
ADORA3 P0DMS8 1/20 0.40
DRD2 P14416 1/20 0.40
ADRA2B P18089 1/20 0.40
ADRA2C P18825 1/20 0.40
DRD1 P21728 1/20 0.40
MC5R P33032 1/20 0.40
OPRM1 P35372 1/20 0.40
DRD3 P35462 1/20 0.40
OPRK1 P41145 1/20 0.40
CCR2 P41597 1/20 0.40
HTR6 P50406 1/20 0.40
SLC6A3 Q01959 1/20 0.40
PDK1 Q15118 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11212437 0.80 PPARA (0.43) ALDH1A1HPGDALOX15HSD17B10CYP1A2
SCHEMBL11210180 0.72 PTGS1 (0.49) ALDH1A1HPGDALOX15HSD17B10TDP1
SCHEMBL10358349 0.72 HPGD (0.58) ALDH1A1HPGDALOX15HSD17B10TDP1
SCHEMBL11207374 0.71 TDP1 (0.43) ALDH1A1HPGDALOX15HSD17B10TDP1
SCHEMBL11211316 0.71 PTGS1 (0.43) ALDH1A1TDP1CYP1A2MAPTHTT
SCHEMBL9357754 0.70 HPGD (0.59) ALDH1A1HPGDALOX15HSD17B10TDP1
SCHEMBL2634521 0.69 HPGD (0.54) ALDH1A1HPGDALOX15HSD17B10TDP1
SCHEMBL10358647 0.69 ALDH1A1 (0.54) ALDH1A1HPGDALOX15HSD17B10TDP1
SCHEMBL9357068 0.68 HPGD (0.56) ALDH1A1HPGDALOX15HSD17B10TDP1
SCHEMBL27404785 0.67 APEX1 (0.51) ALDH1A1HPGDALOX15HSD17B10TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0025262-B1 ALPHA-THIO-ALPHA-ARYL-SUBSTITUTED ALKANONITRILES, PROCESS FOR THEIR PREPARATION, PROCESS FOR PREPARING ALPHA-ARYL-SUBSTITUTED ALKANONITRILES AND THE CORRESPONDING CARBOXYLIC ACIDS THEREFROM AND PROCESS FOR PREPARING INTERMEDIATES SAGAMI CHEMICAL RESEARCH CENTER (JP) 1983-10-05 EP disclosed
US-4340740-A Alpha-thio-alpha-aryl-substituted alkanonitrile and process for preparing alpha-aryl-substituted alkanonitrile therefrom SAGAMI CHEMICAL RESEARCH CENTER (JP) 1982-07-20 US disclosed
EP-0025262-A2 Alpha-thio-alpha-aryl-substituted alkanonitriles, process for their preparation, process for preparing alpha-aryl-substituted alkanonitriles and the corresponding carboxylic acids therefrom and process for preparing intermediates SAGAMI CHEMICAL RESEARCH CENTER (JP) 1981-03-18 EP disclosed