SCHEMBL11207374

SCHEMBL11207374

CC(C#N)(Sc1nc2ccccc2s1)c1cccc(Oc2ccccc2)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
PPARA Q07869 6/20 0.41
THRB P10828 1/20 0.41
RECQL P46063 1/20 0.41
MAPT P10636 6/20 0.40
MEN1 O00255 5/20 0.40
KMT2A Q03164 5/20 0.40
HTT P42858 3/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
TP53 P04637 2/20 0.40
KDM4E B2RXH2 1/20 0.40
JAK2 O60674 1/20 0.40
ATM Q13315 1/20 0.40
ALDH1A1 P00352 1/20 0.39
ADRA2A P08913 1/20 0.39
FBP1 P09467 1/20 0.39
ADORA3 P0DMS8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11210271 0.81 PPARA (0.44) PPARATHRBRECQLMAPTMEN1
SCHEMBL11210711 0.74 AKR1C3 (0.39) TDP1RECQLMAPTMEN1KMT2A
SCHEMBL11208453 0.73 AR (0.39) TDP1L3MBTL1MAPTMEN1KMT2A
SCHEMBL11214020 0.71 ALDH1A1 (0.40) TDP1L3MBTL1PPARAMAPTMEN1
SCHEMBL9353688 0.68 ALDH1A1 (0.59) TDP1L3MBTL1RECQLMAPTMEN1
SCHEMBL11214109 0.68 KMT2A (0.42) TDP1L3MBTL1PPARAMAPTMEN1
SCHEMBL5962402 0.68 ALDH1A1 (0.63) TDP1L3MBTL1RECQLMAPTMEN1
SCHEMBL6576658 0.67 PPARA (0.67) TDP1L3MBTL1PPARARECQLMAPT
SCHEMBL11357018 0.66 MAPT (0.51) TDP1L3MBTL1PPARARECQLMAPT
SCHEMBL13310389 0.66 LTA4H (0.50) MAPTMEN1KMT2ASMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0025262-B1 ALPHA-THIO-ALPHA-ARYL-SUBSTITUTED ALKANONITRILES, PROCESS FOR THEIR PREPARATION, PROCESS FOR PREPARING ALPHA-ARYL-SUBSTITUTED ALKANONITRILES AND THE CORRESPONDING CARBOXYLIC ACIDS THEREFROM AND PROCESS FOR PREPARING INTERMEDIATES SAGAMI CHEMICAL RESEARCH CENTER (JP) 1983-10-05 EP disclosed
US-4340740-A Alpha-thio-alpha-aryl-substituted alkanonitrile and process for preparing alpha-aryl-substituted alkanonitrile therefrom SAGAMI CHEMICAL RESEARCH CENTER (JP) 1982-07-20 US disclosed
EP-0025262-A2 Alpha-thio-alpha-aryl-substituted alkanonitriles, process for their preparation, process for preparing alpha-aryl-substituted alkanonitriles and the corresponding carboxylic acids therefrom and process for preparing intermediates SAGAMI CHEMICAL RESEARCH CENTER (JP) 1981-03-18 EP disclosed