Fluparoxan

Fluparoxan

SCHEMBL112164

Fc1cccc2c1O[C@H]1CNC[C@@H]1O2

nearest known ligand 0.38

Full drug profile on Sugi Atlas →

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 8/20 0.38
CHRNB2 P17787 2/20 0.38
CHRNA4 P43681 2/20 0.38
SLC6A4 P31645 2/20 0.38
SLC6A3 Q01959 2/20 0.38
CA2 P00918 1/20 0.38
HTR6 P50406 4/20 0.36
CHRNA7 P36544 1/20 0.34
HTR1A P08908 6/20 0.34
HTR2C P28335 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.31
ADRA1D P25100 2/20 0.31
ADRA1A P35348 2/20 0.31
ADRA1B P35368 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fluparoxan SCHEMBL9570339 1.00 SLC6A2 (0.38) SLC6A2CHRNB2CHRNA4SLC6A4SLC6A3
Fluparoxan SCHEMBL29401005 1.00 SLC6A2 (0.38) SLC6A2CHRNB2CHRNA4SLC6A4SLC6A3
Fluparoxan SCHEMBL7173629 1.00 SLC6A2 (0.38) SLC6A2CHRNB2CHRNA4SLC6A4SLC6A3
Fluparoxan SCHEMBL9482018 0.98 HTR6 (0.38) SLC6A2CHRNB2CHRNA4SLC6A4SLC6A3
Fluparoxan SCHEMBL122268 0.98 HTR6 (0.38) SLC6A2CHRNB2CHRNA4SLC6A4SLC6A3
Fluparoxan SCHEMBL9482026 0.98 HTR6 (0.38) SLC6A2CHRNB2CHRNA4SLC6A4SLC6A3
SCHEMBL10375117 0.82 BRD4 (0.36) SLC6A2CHRNB2CHRNA4SLC6A4SLC6A3
Hydrochloric Acid SCHEMBL10579193 0.81 BRD4 (0.36) SLC6A2SLC6A4SLC6A3HTR6HTR2C
SCHEMBL10376272 0.81 CHRNB2 (0.34) SLC6A2CHRNB2CHRNA4SLC6A4SLC6A3
SCHEMBL10375154 0.81 CHRNB2 (0.34) SLC6A2CHRNB2CHRNA4SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2020 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3787631-B1 MODULATORS OF ORPHAN NUCLEAR RECEPTORS FOR NASH AND OTHER METABOLIC DISORDERS UNIV EMORY (US) 2025-09-10 EP claimed
EP-3787631-A1 MODULATORS OF ORPHAN NUCLEAR RECEPTORS FOR NASH AND OTHER METABOLIC DISORDERS Emory University (US) 2021-03-10 EP claimed
US-20210052603-A1 MODULATORS OF ORPHAN NUCLEAR RECEPTORS FOR NASH AND OTHER METABOLIC DISORDERS EMORY UNIVERSITY 2021-02-25 US claimed
US-9585884-B2 Pyrimidinone inhibitors of lipoprotein-associated phospholipase A2 AUSPEX PHARMACEUTICALS, INC. (US) 2017-03-07 US claimed
US-20170002015-A1 CYCLOPROPYL MODULATORS OF P2Y12 RECEPTOR AUSPEX PHARMACEUTICALS INC (US) 2017-01-05 US claimed
US-9498481-B2 Cyclopropyl modulators of P2Y12 receptor AUSPEX PHARMACEUTICALS, INC. (US) 2016-11-22 US claimed
US-20160193212-A1 CYCLOPROPYL MODULATORS OF P2Y12 RECEPTOR AUSPEX PHARMACEUTICALS INC (US) 2016-07-07 US claimed
US-9255104-B2 Cyclopropyl modulators of P2Y12 receptor AUSPEX PHARMACEUTICALS, INC. (US) 2016-02-09 US claimed
EP-2961730-A2 METHOD OF MAKING 1-(ACYLOXY)-ALKYL CARBAMATE COMPOUNDS XenoPort, Inc. (US) 2016-01-06 EP claimed
US-20150158809-A9 METHOD OF MAKING 1-(ACYLOXY)-ALKYL CARBAMATE COMPOUNDS XENOPORT, INC. (US) 2015-06-11 US claimed
WO-1997041878-A1 TREATMENT OF MOOD DISORDERS WITH A GROWTH HORMONE SECRETAGOGUE MERCK & CO., INC. (US) 1997-11-13 WO claimed
EP-0532100-A1 Benzodioxinopyrrole derivative as alpha 2-adrenoreceptor antagonist GLAXO GROUP LIMITED (GB) 1993-03-17 EP claimed
EP-0460912-A2 Medicaments for the treatment of sexual disorder GLAXO GROUP LIMITED (GB) 1991-12-11 EP claimed
US-5032603-A Tranquilizers GLAXO GROUP LIMITED (GB) 1991-07-16 US claimed
EP-0407016-A2 Use of benzodioxinopyrrole derivatives in the manufacture of a medicament for the treatment of anxiety GLAXO GROUP LIMITED (GB) 1991-01-09 EP claimed
EP-0162593-B1 HETEROCYCLIC AMINO COMPOUNDS GLAXO GROUP LIMITED (GB) 1990-08-16 EP claimed
EP-0221725-B1 PROCESS FOR PREPARING HETEROCYCLIC COMPOUNDS GLAXO GROUP LIMITED (GB) 1990-08-08 EP claimed
EP-0371793-A2 Use of a benzodioxinopyrrole derivatives for the preparation of a medicament in the treatment of cerebral ischaemia GLAXO GROUP LIMITED (GB) 1990-06-06 EP claimed
US-4880801-A ALPHA 2-ADRENORECEPTOR ANTAGONIST GLAXO GROUP LIMITED (GB) 1989-11-14 US claimed
EP-0221725-A2 Process for preparing heterocyclic compounds GLAXO GROUP LIMITED (GB) 1987-05-13 EP claimed