SCHEMBL1122200

SCHEMBL1122200

COc1cc(-c2ncc(N)nc2N)cc(OC)c1OC

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FYN P06241 10/20 0.53
PIK3CD O00329 1/20 0.47
ABL1 P00519 1/20 0.47
EGFR P00533 1/20 0.47
HCK P08631 1/20 0.47
SRC P12931 1/20 0.47
KDR P35968 1/20 0.47
PIK3CA P42336 1/20 0.47
PIK3CB P42338 1/20 0.47
MTOR P42345 1/20 0.47
PIK3CG P48736 1/20 0.47
EPHB4 P54760 1/20 0.47
PRKDC P78527 1/20 0.47
PI4KB Q9UBF8 1/20 0.47
NEK2 P51955 2/20 0.46
TSHR P16473 2/20 0.45
KDM4E B2RXH2 1/20 0.45
POLB P06746 1/20 0.45
GAA P10253 1/20 0.45
TGFBR1 P36897 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28855953 0.78 FYN (0.53) FYNPIK3CDABL1EGFRHCK
SCHEMBL29870262 0.75 KDM4E (0.50) FYNTSHRKDM4EPOLBMEN1
SCHEMBL975873 0.75 KDM4E (0.50) FYNTSHRKDM4EPOLBMEN1
SCHEMBL6722240 0.73 KMT2A (0.55) PIK3CDABL1EGFRHCKSRC
SCHEMBL20589749 0.72 FYN (0.50) FYNTSHRKDM4EPOLBGAA
SCHEMBL28901285 0.71 TUBB4A (0.47) FYNADORA2AADORA1
SCHEMBL27612599 0.71 ADORA2A (0.53) FYNPIK3CDABL1EGFRHCK
SCHEMBL2437579 0.71 DHFR (0.67) FYNTSHRGAATGFBR1MEN1
SCHEMBL20589457 0.70 ABL1 (0.64) FYNABL1TGFBR1CHEK2
SCHEMBL30268270 0.70 PIK3CD (0.49) FYNPIK3CDABL1EGFRHCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1831184-B1 PYRAZINES AND PYRIDINES AND DERIVATIVES THEREOF AS THERAPEUTIC COMPOUNDS WELLCOME TRUST LTD (GB) 2011-02-09 EP disclosed