SCHEMBL11222341

SCHEMBL11222341

Clc1ncc(OCc2ccccc2)nc1N1CCOCC1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 1/20 0.61
ALDH1A1 P00352 5/20 0.55
TSHR P16473 4/20 0.55
HSD17B10 Q99714 3/20 0.55
ALOX15 P16050 1/20 0.55
MAPK1 P28482 1/20 0.55
SMN1; SMN2 Q16637 1/20 0.48
PRMT5 O14744 3/20 0.47
MGMT P16455 1/20 0.47
KDM4E B2RXH2 3/20 0.45
GAA P10253 1/20 0.45
PKM P14618 1/20 0.45
CNR1 P21554 1/20 0.44
CNR2 P34972 1/20 0.44
LMNA P02545 2/20 0.43
THRB P10828 1/20 0.43
PDE4A P27815 1/20 0.43
PDE4B Q07343 1/20 0.43
PDE4C Q08493 1/20 0.43
PDE4D Q08499 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11220678 0.85 CYP11B2 (0.61) CYP11B2ALDH1A1TSHRHSD17B10ALOX15
SCHEMBL11218413 0.82 POLB (0.50) CYP11B2ALDH1A1TSHRHSD17B10KDM4E
SCHEMBL18489956 0.76 CYP11B2 (1.00) CYP11B2ALDH1A1TSHRHSD17B10ALOX15
SCHEMBL10414485 0.75 CYP11B2 (0.58) CYP11B2ALDH1A1TSHRHSD17B10ALOX15
SCHEMBL3990390 0.75 CYP11B2 (0.65) CYP11B2ALDH1A1TSHRHSD17B10ALOX15
SCHEMBL11229317 0.75 NOS1 (0.58) ALDH1A1TSHRHSD17B10MAPK1SMN1; SMN2
SCHEMBL25230198 0.74 CYP11B2 (0.60) CYP11B2ALDH1A1TSHRHSD17B10ALOX15
Hydrochloric Acid SCHEMBL6284101 0.73 HTR2C (0.70)
SCHEMBL7712443 0.72 MGMT (0.58) CYP11B2ALDH1A1TSHRHSD17B10ALOX15
SCHEMBL8131727 0.72 MGMT (0.53) CYP11B2ALDH1A1TSHRHSD17B10ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4343802-A ADRENERGIC BLOCKING, ANTIARRYHYTHMIA, AND CARDIOTONIC AGENTS MERCK, SHARP & DOHME (I.A.) CORP. (US) 1982-08-10 US disclosed
US-4193995-A B-ADRENERGIC BLOCKING AGENTS MERCK SHARP & DOHME (I.A.) CORP. (US) 1980-03-18 US disclosed
US-4042586-A ADRENERGIC BLOCKING AGENTS MERCK SHARP & DOHME (I.A.) CORPORATION (US) 1977-08-16 US disclosed
US-3946009-A ADRENERGIC BLOCKING AGENTS MERCK SHARP & DOHME (I.A.) CORPORATION (US) 1976-03-23 US disclosed