SCHEMBL11229317

SCHEMBL11229317

Clc1ncc(-c2ccccc2)nc1N1CCOCC1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 1/20 0.58
ALDH1A1 P00352 2/20 0.55
ADK P55263 1/20 0.53
MTOR P42345 2/20 0.52
HSD17B10 Q99714 2/20 0.50
CASP1 P29466 1/20 0.50
TRPM8 Q7Z2W7 1/20 0.49
MAPK1 P28482 2/20 0.49
MAPT P10636 2/20 0.49
TSHR P16473 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
AR P10275 1/20 0.49
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
POLB P06746 1/20 0.47
ROCK2 O75116 1/20 0.47
ROCK1 Q13464 1/20 0.47
GAA P10253 1/20 0.47
ABL1 P00519 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11223817 0.83 NOS1 (0.65) NOS1ALDH1A1ADKMTORHSD17B10
SCHEMBL11218413 0.77 POLB (0.50) ALDH1A1MTORHSD17B10CASP1TRPM8
SCHEMBL11148029 0.75 ALDH1A1 (0.48) ALDH1A1ADKHSD17B10MAPK1TSHR
SCHEMBL11225591 0.75 KDM4E (0.45) ALDH1A1ADKMAPK1MAPTTSHR
SCHEMBL11222341 0.75 CYP11B2 (0.61) ALDH1A1HSD17B10CASP1TRPM8MAPK1
SCHEMBL14725974 0.74 ALDH1A1 (0.48) ALDH1A1ADKMTORMAPK1MAPT
SCHEMBL11218532 0.74 PIK3CA (0.47) ALDH1A1ADKMTORMAPK1MAPT
SCHEMBL5317835 0.74 NOS1 (1.00) NOS1ALDH1A1ADKMTORHSD17B10
Water SCHEMBL6491267 0.73 NOS1 (0.98) NOS1ALDH1A1ADKMTORHSD17B10
SCHEMBL1752981 0.72 ALDH1A1 (0.55) ALDH1A1MTORHSD17B10CASP1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4343802-A ADRENERGIC BLOCKING, ANTIARRYHYTHMIA, AND CARDIOTONIC AGENTS MERCK, SHARP & DOHME (I.A.) CORP. (US) 1982-08-10 US disclosed
US-4193995-A B-ADRENERGIC BLOCKING AGENTS MERCK SHARP & DOHME (I.A.) CORP. (US) 1980-03-18 US disclosed
US-4042586-A ADRENERGIC BLOCKING AGENTS MERCK SHARP & DOHME (I.A.) CORPORATION (US) 1977-08-16 US disclosed
US-3946009-A ADRENERGIC BLOCKING AGENTS MERCK SHARP & DOHME (I.A.) CORPORATION (US) 1976-03-23 US disclosed