SCHEMBL11222599

SCHEMBL11222599

O=C1CCCC(=O)C1c1c(Br)ccc(Cl)c1F

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 9/20 0.35
HTR2C P28335 9/20 0.35
HTR2B P41595 4/20 0.35
IL1RN P18510 1/20 0.32
ERAP2 Q6P179 1/20 0.32
ERAP1 Q9NZ08 1/20 0.32
USP2 O75604 1/20 0.30
HPGD P15428 1/20 0.30
KDM1A O60341 2/20 0.30
KCNH2 Q12809 2/20 0.30
KDM1B Q8NB78 2/20 0.30
ABCC9 O60706 1/20 0.30
ABCC8 Q09428 1/20 0.30
KCNJ11 Q14654 1/20 0.30
KCNJ8 Q15842 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11227830 0.68 HSD11B1 (0.34) IL1RNERAP2ERAP1
SCHEMBL11224580 0.66 TDP1 (0.33) IL1RNERAP2ERAP1
SCHEMBL11227905 0.65 CYP3A4 (0.39)
SCHEMBL2014602 0.64 KDM1A (0.39) USP2HPGDKDM1AKCNH2KDM1B
SCHEMBL31342136 0.64 KDM1A (0.39) USP2HPGDKDM1AKCNH2KDM1B
SCHEMBL11229583 0.64 HCRTR1 (0.39)
SCHEMBL23674528 0.63 CDC7 (0.36) KDM1AKCNH2KDM1B
SCHEMBL11891671 0.62 EPAS1 (0.34) HTR2AHTR2CHTR2BKDM1AKCNH2
SCHEMBL30223191 0.62 HTR2A (0.32) HTR2AHTR2CHTR2B
SCHEMBL15821759 0.62 CA1 (0.35) HTR2AHTR2CHTR2BUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0007243-B1 2-ARYL-1,3-CYCLOHEXANEDIONE COMPOUNDS AND ALKALI METAL SALTS, AMMONIUM SALTS AND ENOL ESTERS THEREOF, COMPOSITION AND METHOD OF CONTROLLING ACARINA ECTOPARASITES ON WARMBLOODED ANIMALS UNION CARBIDE CORPORATION (US) 1982-11-17 EP disclosed
US-4257858-A REACTING A CYCLOHEXA-1,3-DIONE-2-DIAZIDE WITH AN ARYL COMPOUND UNION CARBIDE CORPORATION (US) 1981-03-24 US disclosed
US-4256657-A CYCLIZATION, ACID CATALYST UNION CARBIDE CORPORATION (US) 1981-03-17 US disclosed
US-4256658-A CYCLIZATION, BASIC CATALYST UNION CARBIDE CORPORATION (US) 1981-03-17 US disclosed
US-4256659-A Method of preparing 2-aryl-1,3-cyclohexanedione compounds UNION CARBIDE CORPORATION (US) 1981-03-17 US disclosed
US-4209532-A Biocidal 2-aryl-1,3-cyclohexane dione compounds and alkali metal and ammonium salts thereof UNION CARBIDE CORPORATION (US) 1980-06-24 US disclosed
EP-0007243-A1 2-Aryl-1,3-cyclohexanedione compounds and alkali metal salts, ammonium salts and enol esters thereof, composition and method of controlling acarina ectoparasites on warmblooded animals UNION CARBIDE CORPORATION (US) 1980-01-23 EP disclosed
US-4175135-A Method of controlling acarina ectoparasites on warmblooded animals by orally administering to the animal an ectoparasitically effective amount of a 2-aryl-1,3-cyclohexanedione compound, and alkali metal salts, ammonium salts and enol esters thereof UNION CARBIDE CORPORATION (US) 1979-11-20 US disclosed