SCHEMBL11222772

SCHEMBL11222772

CC(C)c1nc(Br)cnc1Br

nearest known ligand 0.31

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.31
PAK4 O96013 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13396971 0.82 MAPK1 (0.31) MAPK1
SCHEMBL25946352 0.80 MAPK1 (0.31) MAPK1
SCHEMBL10925572 0.80 PAK4 (0.31) PAK4
SCHEMBL11221495 0.78 GABRA1 (0.30)
SCHEMBL25928367 0.76 MAPK1 (0.31) MAPK1
SCHEMBL16248170 0.74 DHFR (0.31)
SCHEMBL25928446 0.72
SCHEMBL25928457 0.72 JAK2 (0.36) PAK4
SCHEMBL17423958 0.72 ALDH1A1 (0.41)
SCHEMBL31281424 0.69

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4343802-A ADRENERGIC BLOCKING, ANTIARRYHYTHMIA, AND CARDIOTONIC AGENTS MERCK, SHARP & DOHME (I.A.) CORP. (US) 1982-08-10 US disclosed
US-4193995-A B-ADRENERGIC BLOCKING AGENTS MERCK SHARP & DOHME (I.A.) CORP. (US) 1980-03-18 US disclosed
US-4042586-A ADRENERGIC BLOCKING AGENTS MERCK SHARP & DOHME (I.A.) CORPORATION (US) 1977-08-16 US disclosed
US-3946009-A ADRENERGIC BLOCKING AGENTS MERCK SHARP & DOHME (I.A.) CORPORATION (US) 1976-03-23 US disclosed