SCHEMBL11223736

SCHEMBL11223736

CCCN1CC(C(C#N)(c2ccccc2)c2ccccc2)C1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KCNA3 P22001 5/20 0.42
RAB9A P51151 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
DRD2 P14416 3/20 0.40
DRD1 P21728 1/20 0.40
DRD4 P21917 1/20 0.40
DRD5 P21918 1/20 0.40
DRD3 P35462 1/20 0.40
CHRM2 P08172 1/20 0.40
CHRM1 P11229 1/20 0.40
CHRM3 P20309 1/20 0.40
SIGMAR1 Q99720 1/20 0.38
CCR1 P32246 1/20 0.38
OPRM1 P35372 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11220493 0.91 CCR1 (0.44) KCNA3RAB9ANPSR1CHRM2CHRM1
SCHEMBL11226666 0.88 KCNA3 (0.40) KCNA3RAB9ANPSR1DRD2DRD4
SCHEMBL11225253 0.84 SLC6A3 (0.44) KCNA3DRD2DRD3CHRM3SIGMAR1
SCHEMBL11228398 0.82 ATM (0.44) KCNA3RAB9ANPSR1DRD2DRD4
SCHEMBL11234010 0.81 CYP3A4 (0.39) KCNA3RAB9ANPSR1CHRM2CHRM1
SCHEMBL11235320 0.80 KCNA3 (0.50) KCNA3DRD2DRD3SIGMAR1OPRM1
SCHEMBL14125383 0.79 KCNA3 (0.46) KCNA3OPRM1
SCHEMBL14029031 0.79 KCNA3 (0.46) KCNA3OPRM1
SCHEMBL2619538 0.79 KCNA3 (0.46) KCNA3OPRM1
SCHEMBL11220612 0.75 CYP2D6 (0.41) KCNA3RAB9ANPSR1DRD2DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4324791-A DERIVATIVES OF 3,3-DIPHENYL-2-PYRROLIDINONES A. H. ROBINS COMPANY, INC. (US) 1982-04-13 US disclosed
US-4296037-A 4,5-Dihydro-3,3-diphenyl-4-hydrocarbylaminomethylfuran-2(3H) ones A. H. ROBINS COMPANY, INCORPORATED (US) 1981-10-20 US disclosed
US-4144245-A 4-Hydroxymethyl-2-pyrrolidinones A. H. ROBINS COMPANY, INC. (US) 1979-03-13 US disclosed
US-4120969-A ANALGETIC, ANTIDIARRHEAL ACTIVITY A. H. ROBINS COMPANY, INCORPORATED (US) 1978-10-17 US disclosed
US-4119637-A 4-Hydroxymethyl-2-pyrrolidinones A. H. ROBINS COMPANY, INC. (US) 1978-10-10 US disclosed