SCHEMBL11234010

SCHEMBL11234010

CC(C)CN1CC(C(C#N)(c2ccccc2)c2ccccc2)C1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.39
CYP2D6 P10635 2/20 0.39
CHRM2 P08172 2/20 0.39
CHRM1 P11229 2/20 0.39
CHRM3 P20309 2/20 0.39
CYP2C19 P33261 1/20 0.39
KCNA3 P22001 6/20 0.38
RAB9A P51151 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
HRH3 Q9Y5N1 2/20 0.35
MEN1 O00255 3/20 0.34
PIK3CD O00329 1/20 0.33
KMT2A Q03164 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11732329 0.89 KCNA3 (0.43) CYP3A4CYP2D6CHRM2CHRM1CHRM3
SCHEMBL11226666 0.83 KCNA3 (0.40) CYP3A4CYP2D6CHRM2CHRM1CHRM3
SCHEMBL11223736 0.81 KCNA3 (0.42) CHRM2CHRM1CHRM3KCNA3RAB9A
SCHEMBL11220612 0.80 CYP2D6 (0.41) CYP3A4CYP2D6CHRM2CHRM1CHRM3
SCHEMBL11235320 0.79 KCNA3 (0.50) KCNA3
SCHEMBL11220493 0.78 CCR1 (0.44) CHRM2CHRM1CHRM3KCNA3RAB9A
SCHEMBL11228398 0.78 ATM (0.44) CYP3A4CYP2D6CHRM2CHRM1CHRM3
SCHEMBL11832937 0.78 MEN1 (0.40) CHRM2CHRM1CHRM3KCNA3MEN1
SCHEMBL11226664 0.77 CYP2D6 (0.46) CYP3A4CYP2D6CHRM2CHRM1CHRM3
SCHEMBL11225253 0.77 SLC6A3 (0.44) CHRM3KCNA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4324791-A DERIVATIVES OF 3,3-DIPHENYL-2-PYRROLIDINONES A. H. ROBINS COMPANY, INC. (US) 1982-04-13 US disclosed
US-4296037-A 4,5-Dihydro-3,3-diphenyl-4-hydrocarbylaminomethylfuran-2(3H) ones A. H. ROBINS COMPANY, INCORPORATED (US) 1981-10-20 US disclosed
US-4144245-A 4-Hydroxymethyl-2-pyrrolidinones A. H. ROBINS COMPANY, INC. (US) 1979-03-13 US disclosed
US-4120969-A ANALGETIC, ANTIDIARRHEAL ACTIVITY A. H. ROBINS COMPANY, INCORPORATED (US) 1978-10-17 US disclosed
US-4119637-A 4-Hydroxymethyl-2-pyrrolidinones A. H. ROBINS COMPANY, INC. (US) 1978-10-10 US disclosed