SCHEMBL11226052

SCHEMBL11226052

ClCCOCC1OCCCc2cc3c(cc21)OCO3

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.34
HSD17B10 Q99714 3/20 0.34
ALDH1A1 P00352 2/20 0.34
GLA P06280 2/20 0.34
HPGD P15428 2/20 0.34
CASP1 P29466 2/20 0.34
CASP7 P55210 2/20 0.34
CYP2D6 P10635 1/20 0.34
CHRNA7 P36544 3/20 0.34
DRD1 P21728 3/20 0.33
DRD2 P14416 2/20 0.33
ADRA1A P35348 1/20 0.33
GAA P10253 1/20 0.33
HTR1A P08908 1/20 0.32
CYP3A4 P08684 1/20 0.32
MAPT P10636 1/20 0.32
MAPK13 O15264 1/20 0.32
MAPK12 P53778 1/20 0.32
MAPK11 Q15759 1/20 0.32
MAPK14 Q16539 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11220977 0.83 KDM4E (0.38) KDM4EHSD17B10ALDH1A1GLAHPGD
SCHEMBL11217894 0.80 MAOA (0.36) KDM4EALDH1A1CHRNA7
SCHEMBL11226631 0.77 KDM4E (0.39) KDM4EHSD17B10ALDH1A1GLAHPGD
SCHEMBL11232820 0.77 CHRNA7 (0.33) KDM4EHSD17B10ALDH1A1GLAHPGD
SCHEMBL11232660 0.76 ALDH1A1 (0.39) ALDH1A1CYP2D6DRD2GAAHTR1A
SCHEMBL11222512 0.76 HTR2C (0.40) KDM4EALDH1A1CYP3A4MAPT
SCHEMBL11226050 0.75
SCHEMBL11219842 0.75 MEN1 (0.36) MAPT
SCHEMBL11223974 0.75 HTR2A (0.42) KDM4EALDH1A1HTR1A
SCHEMBL11225616 0.74 KDM4E (0.39) KDM4EHSD17B10ALDH1A1GLAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4352805-A BENZOXEPINE DERIVATIVES THE UPJOHN COMPANY (US) 1982-10-05 US disclosed
US-4312868-A HYPOTENSIVE, ANTIPSYCHOTIC THE UPJOHN COMPANY (US) 1982-01-26 US disclosed
US-4251526-A HYPOTENSIVE AGENTS AND ANTIPSYCHOTIC PHARMACIA & UPJOHN COMPANY 1981-02-17 US disclosed
US-4250181-A HYPOTENSIVE AGENTS, ANTIDEPRESSANTS THE UPJOHN COMPANY (US) 1981-02-10 US disclosed
US-4250175-A HYPOTENSIVE AGENTS, ANTIDEPRESSANTS PHARMACIA & UPJOHN COMPANY 1981-02-10 US disclosed
US-4247553-A HYPOTENSIVE AGENTS, ANTIDEPRESSANTS THE UPJOHN COMPANY (US) 1981-01-27 US disclosed
US-4179510-A ISOCHROMANS AND 2-BENZOXEPINS THE UPJOHN COMPANY (US) 1979-12-18 US disclosed
US-4166062-A HYPOTENSIVE AGENTS, CNS, ANTIDEPRESSANTS THE UPJOHN COMPANY (US) 1979-08-28 US disclosed
US-4153612-A 2-Benzoxepins THE UPJOHN COMPANY (US) 1979-05-08 US disclosed