SCHEMBL11227397

SCHEMBL11227397

COc1ccc2c(C)cc(=O)oc2c1N

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 6/20 0.72
KDM4E B2RXH2 6/20 0.72
ALDH1A1 P00352 6/20 0.72
HPGD P15428 4/20 0.72
TSHR P16473 2/20 0.72
L3MBTL1 Q9Y468 1/20 0.72
MCL1 Q07820 2/20 0.68
GAA P10253 5/20 0.63
GFER P55789 1/20 0.63
MAOA P21397 2/20 0.56
ALPL P05186 3/20 0.52
CYP1A2 P05177 2/20 0.52
LMNA P02545 4/20 0.50
MAPT P10636 4/20 0.50
KMT2A Q03164 3/20 0.50
MAPK1 P28482 2/20 0.50
MAOB P27338 2/20 0.50
ALPI P09923 1/20 0.50
GLA P06280 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9463878 0.84 ALDH1A1 (1.00) HSD17B10KDM4EALDH1A1HPGDTSHR
SCHEMBL4772250 0.83 KDM4E (0.74) HSD17B10KDM4EALDH1A1HPGDTSHR
SCHEMBL15984891 0.81 MCL1 (1.00) HSD17B10KDM4EALDH1A1HPGDTSHR
SCHEMBL5321909 0.81 KDM4E (0.72) HSD17B10KDM4EALDH1A1HPGDTSHR
SCHEMBL18232224 0.80 KDM4E (0.70) HSD17B10KDM4EALDH1A1HPGDTSHR
Trimethylammonium SCHEMBL9481220 0.79 ALDH1A1 (0.88) HSD17B10KDM4EALDH1A1HPGDTSHR
SCHEMBL11227296 0.78 MCL1 (0.68) HSD17B10KDM4EALDH1A1HPGDTSHR
SCHEMBL8724340 0.78 GAA (1.00) HSD17B10KDM4EALDH1A1HPGDMCL1
SCHEMBL22902127 0.77 ALDH1A1 (0.42) HSD17B10KDM4EALDH1A1HPGDTSHR
SCHEMBL11195848 0.76 KDM4E (0.74) HSD17B10KDM4EALDH1A1HPGDTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4309353-A ANTI-ALLERGIC AGENTS CIBA-GEIGY CORPORATION (US) 1982-01-05 US disclosed
US-4205082-A ANTI-ALLERGIC AGENTS CIBA-GEIGY CORPORATION (US) 1980-05-27 US disclosed