SCHEMBL11229145

SCHEMBL11229145

CC(=O)C=CNc1cc(-c2cccnc2)c[nH]c1=O

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TTK P33981 4/20 0.51
AURKB Q96GD4 3/20 0.51
INCENP Q9NQS7 3/20 0.51
AURKA O14965 2/20 0.51
ITK Q08881 7/20 0.42
MKNK1 Q9BUB5 2/20 0.41
MKNK2 Q9HBH9 2/20 0.41
PDPK1 O15530 1/20 0.41
AKT2 P31751 1/20 0.41
NR4A2 P43354 1/20 0.40
KIT P10721 2/20 0.39
SRC P12931 2/20 0.39
FLT3 P36888 2/20 0.39
KMO O15229 1/20 0.39
GPR142 Q7Z601 4/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11229132 1.00 TTK (0.51) TTKAURKBINCENPAURKAITK
SCHEMBL11222397 0.85 ITK (0.55) TTKAURKBINCENPAURKAITK
SCHEMBL11222394 0.85 ITK (0.55) TTKAURKBINCENPAURKAITK
SCHEMBL11233683 0.82 ITK (0.41) TTKAURKBINCENPAURKAITK
SCHEMBL11233679 0.82 ITK (0.41) TTKAURKBINCENPAURKAITK
SCHEMBL11234330 0.81 TTK (0.51) TTKAURKBINCENPAURKAITK
SCHEMBL11234332 0.81 TTK (0.51) TTKAURKBINCENPAURKAITK
SCHEMBL11219764 0.80 CCNC (0.51) TTKAURKBINCENPAURKAITK
SCHEMBL11219760 0.80 CCNC (0.51) TTKAURKBINCENPAURKAITK
SCHEMBL11228274 0.80 MKNK1 (0.39) TTKAURKBINCENPAURKAITK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4362735-A 3-[(3-Oxo-1-butenyl)amino]-5-(pyridinyl)-2(1H)-pyridinones and their cardiotonic use STERLING DRUG INC. (US) 1982-12-07 US disclosed