SCHEMBL11233683

SCHEMBL11233683

CC(=O)C=CNc1cc(-c2cncc(C)c2)c[nH]c1=O

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ITK Q08881 8/20 0.41
GPR142 Q7Z601 7/20 0.39
TTK P33981 4/20 0.37
KIT P10721 3/20 0.37
SRC P12931 3/20 0.37
FLT3 P36888 3/20 0.37
AURKB Q96GD4 3/20 0.37
INCENP Q9NQS7 3/20 0.37
AURKA O14965 2/20 0.36
PIK3CG P48736 1/20 0.34
PRMT5 O14744 1/20 0.32
WDR77 Q9BQA1 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11233679 1.00 ITK (0.41) ITKGPR142TTKKITSRC
SCHEMBL11229145 0.82 TTK (0.51) ITKGPR142TTKKITSRC
SCHEMBL11229132 0.82 TTK (0.51) ITKGPR142TTKKITSRC
SCHEMBL11222394 0.81 ITK (0.55) ITKGPR142TTKKITSRC
SCHEMBL11222397 0.81 ITK (0.55) ITKGPR142TTKKITSRC
SCHEMBL11223826 0.81 ITK (0.39) ITKGPR142TTKKITSRC
SCHEMBL11228964 0.81 ITK (0.46) ITKGPR142TTKKITSRC
SCHEMBL11228960 0.81 ITK (0.46) ITKGPR142TTKKITSRC
SCHEMBL11449526 0.76 ITK (0.40) ITKGPR142TTKKITSRC
SCHEMBL11219764 0.74 CCNC (0.51) ITKGPR142TTKKITSRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4362735-A 3-[(3-Oxo-1-butenyl)amino]-5-(pyridinyl)-2(1H)-pyridinones and their cardiotonic use STERLING DRUG INC. (US) 1982-12-07 US disclosed