SCHEMBL11230744

SCHEMBL11230744

COCCn1c(=S)[nH]c2cc(-c3ccncc3)cnc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 1/20 0.46
PKM P14618 2/20 0.45
POLB P06746 1/20 0.45
ALDH1A1 P00352 8/20 0.44
MAPK1 P28482 1/20 0.44
HSD17B10 Q99714 3/20 0.44
KDM4E B2RXH2 2/20 0.43
USP2 O75604 1/20 0.43
GAA P10253 1/20 0.43
CASP1 P29466 1/20 0.43
CASP7 P55210 1/20 0.43
CYP1A2 P05177 2/20 0.40
CYP2C19 P33261 2/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
RXFP1 Q9HBX9 1/20 0.40
HPGD P15428 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
PDE3B Q13370 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11157976 0.86 ALDH1A1 (0.50) PKMPOLBALDH1A1HSD17B10KDM4E
SCHEMBL11225776 0.84 PDE3B (0.43) ALDH1A1CYP1A2CYP2C19MEN1KMT2A
SCHEMBL11336866 0.81 PDE3B (0.50) POLBMEN1KMT2ANPSR1RXFP1
Water SCHEMBL11233745 0.79 PDE3B (0.49) POLBMEN1KMT2APDE3BPDE3A
Water SCHEMBL11233741 0.79 PDE3B (0.49) POLBMEN1KMT2APDE3BPDE3A
SCHEMBL11241051 0.79 ALDH1A1 (0.48) PKMALDH1A1HSD17B10KDM4EGAA
SCHEMBL11233887 0.78 PDE3B (0.38) PDE3BPDE3APDE4BKDR
SCHEMBL11233166 0.77 RAB9A (0.47) RAB9APKMPOLBALDH1A1MAPK1
SCHEMBL11381432 0.71 AXL (0.40) ALDH1A1MAPK1HSD17B10KDM4EGAA
SCHEMBL11157645 0.71 PDE3B (0.49) CYP1A2MEN1KMT2ASMN1; SMN2PDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4309537-A Production of imidazo[4,5-b]pyridin-2-ones or thiones STERLING DRUG INC. (US) 1982-01-05 US disclosed
US-4297360-A 5-(Pyridinyl)pyridine-2,3-diamines, preparation thereof and their cardiotonic use STERLING DRUG INC. (US) 1981-10-27 US disclosed
US-4294837-A 1,3-Dihydro-6-(pyridinyl)-2H-imidazo[4,5-b]pyridin-2-ones and -imidazo[4,5-b]pyridine-2-thiones and their cardiotonic use STERLING DRUG INC. (US) 1981-10-13 US disclosed