SCHEMBL11233117

SCHEMBL11233117

CCCOC(=O)c1cc(-c2cccnc2)c(C)[nH]c1=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.47
LMNA P02545 5/20 0.47
L3MBTL1 Q9Y468 2/20 0.47
MAPT P10636 2/20 0.47
MMP2 P08253 1/20 0.45
MMP13 P45452 1/20 0.45
MMP14 P50281 1/20 0.45
CDK5 Q00535 1/20 0.44
CDK5R1 Q15078 1/20 0.44
KDM4E B2RXH2 5/20 0.43
DCTPP1 Q9H773 1/20 0.43
HSD17B10 Q99714 1/20 0.43
GAA P10253 3/20 0.42
HPGD P15428 1/20 0.42
NPC1 O15118 2/20 0.42
RAB9A P51151 1/20 0.42
POLB P06746 3/20 0.41
MEN1 O00255 1/20 0.41
MAPK1 P28482 1/20 0.41
HTT P42858 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11236586 0.81 CDK5 (0.53) ALDH1A1LMNAL3MBTL1MAPTMMP2
SCHEMBL11236769 0.80 KDM4E (0.50) LMNAKDM4EHSD17B10GAAHPGD
SCHEMBL11078693 0.79 MKNK1 (0.56) LMNAKMT2A
SCHEMBL11242636 0.78 CDK5 (0.62) ALDH1A1LMNAL3MBTL1MAPTCDK5
SCHEMBL2673559 0.76 ALK (0.47) ALDH1A1LMNAMMP2MMP13MMP14
SCHEMBL11229029 0.75 ALK (0.43) ALDH1A1LMNAKDM4EHSD17B10HPGD
SCHEMBL11229059 0.74 MKNK1 (0.43) ALDH1A1LMNAKDM4EHSD17B10HPGD
SCHEMBL4428979 0.73 ALK (0.53) ALDH1A1L3MBTL1MAPTMMP2MMP13
SCHEMBL5903422 0.72 CDK5 (0.80) CDK5CDK5R1
SCHEMBL11229727 0.72 PDE3B (0.68) ALDH1A1LMNAKDM4EHSD17B10HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4312875-A 5-(Pyridinyl)-6-(lower-alkyl)-2(1H)-pyridinones, 1,2-dihydro-2-oxo-5-(pyridinyl)-6-(lower-alkyl)nicotinic acids and lower-alkyl esters thereof, and cardiotonic use thereof STERLING DRUG INC. (US) 1982-01-26 US disclosed