SCHEMBL11229029

SCHEMBL11229029

Cc1[nH]c(=O)c(C(=N)NO)cc1-c1cccnc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 1/20 0.43
KMT2A Q03164 1/20 0.42
PIK3C3 Q8NEB9 1/20 0.41
PDE3B Q13370 3/20 0.41
PDE3A Q14432 3/20 0.41
AURKB Q96GD4 1/20 0.41
INCENP Q9NQS7 1/20 0.41
CYP2A6 P11509 1/20 0.40
HDAC3 O15379 1/20 0.40
HDAC4 P56524 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC7 Q8WUI4 1/20 0.40
HDAC2 Q92769 1/20 0.40
HDAC10 Q969S8 1/20 0.40
HDAC11 Q96DB2 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
HDAC9 Q9UKV0 1/20 0.40
HDAC5 Q9UQL6 1/20 0.40
PDE4A P27815 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11230843 0.85 PDE3B (0.57) PDE3BPDE3AAURKBINCENPPDE4A
SCHEMBL11233012 0.84 PDE3B (0.42) KMT2APDE3BPDE3ACYP2A6HDAC3
SCHEMBL11236769 0.83 KDM4E (0.50) ALKKMT2APDE3BPDE3AAURKB
SCHEMBL11078693 0.82 MKNK1 (0.56) ALKKMT2APDE3BPDE3AAURKB
SCHEMBL11229059 0.79 MKNK1 (0.43) ALKKMT2APIK3C3PDE3BPDE3A
SCHEMBL11243997 0.77 ALK (0.46) ALKKMT2APIK3C3PDE3BPDE3A
SCHEMBL11229727 0.77 PDE3B (0.68) ALKKMT2APIK3C3PDE3BPDE3A
SCHEMBL11238459 0.77 ALK (0.48) ALKKMT2APIK3C3PDE3BPDE3A
SCHEMBL2673559 0.76 ALK (0.47) ALKKMT2APIK3C3PDE3BPDE3A
SCHEMBL11233117 0.75 ALDH1A1 (0.47) KMT2AKDM4EHPGDALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4339584-A Process for preparing 3-amino-5-(pyridinyl)-2(1H)-pyridinones via N-hydroxy-1,2-dihydro-2-oxo-5-(pyridinyl)-nicotinimidamide by reaction with polyphosphoric acid STERLING DRUG INC. (US) 1982-07-13 US disclosed
US-4305948-A N-Hydroxy-1,2-dihydro-2-oxo-5-(pyridinyl)-nicotinimidamide and their cardiotonic use STERLING DRUG INC. (US) 1981-12-15 US disclosed