SCHEMBL11233899

SCHEMBL11233899

OCCc1ccc2c(c1)sc1ccc(Cl)cc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.41
CHRNA7 P36544 1/20 0.40
MAPT P10636 2/20 0.37
ALDH1A1 P00352 1/20 0.37
ALOX5 P09917 1/20 0.37
GAA P10253 1/20 0.37
BACE1 P56817 1/20 0.37
BCKDK O14874 1/20 0.36
MCL1 Q07820 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
CYP2A6 P11509 2/20 0.34
AKR1B1 P15121 1/20 0.34
KEAP1 Q14145 1/20 0.34
NFE2L2 Q16236 1/20 0.34
ROCK1 Q13464 1/20 0.33
SLC22A12 Q96S37 1/20 0.33
PYGL P06737 1/20 0.33
IDO1 P14902 1/20 0.33
IGF1R P08069 1/20 0.33
ALOX15 P16050 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11240017 0.79 KEAP1 (0.51) KDM4EMAPTALDH1A1GAABCKDK
SCHEMBL11253511 0.79 KDM4E (0.42) KDM4EMAPTGAABCKDKMCL1
Methane SCHEMBL11235653 0.78 KEAP1 (0.50) KDM4EMAPTALDH1A1GAABCKDK
SCHEMBL11232073 0.78 SIRT1 (0.44) KDM4EMAPTALDH1A1BCKDKMCL1
SCHEMBL18903328 0.77 GPR3 (0.50) KDM4EMAPTALDH1A1ALOX5GAA
Methane SCHEMBL11235493 0.77 SIRT1 (0.43) KDM4EMAPTALDH1A1BCKDKMCL1
SCHEMBL11250520 0.76 CYP4F2 (0.47) KDM4ESLC22A12ALOX15
SCHEMBL2308278 0.76 KDM4E (0.41) KDM4EMAPTALDH1A1ALOX5GAA
SCHEMBL3258493 0.75 KDM4E (0.61) KDM4ECHRNA7MAPTALDH1A1GAA
SCHEMBL24343656 0.75 KDM4E (0.46) KDM4EMAPTBCKDKMCL1RXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4334078-A ANTIINFLAMMATORY AGENTS, ANALGESICS, ANTIRHEUMATICS HOFFMANN-LA ROCHE INC. (US) 1982-06-08 US disclosed
US-4219657-A USED AS ANTIINFLAMATORY AGENTS, ANALGESICS, ANTIRHEUMATIC AGENTS HOFFMANN-LA ROCHE INC. (US) 1980-08-26 US disclosed