SCHEMBL11234003

SCHEMBL11234003

CCc1cccc(C(=O)O)c1N=Cc1ccc(Cl)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.41
CLCN2 P51788 1/20 0.40
TRPA1 O75762 1/20 0.39
MRGPRX4 Q96LA9 4/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
NR4A1 P22736 1/20 0.39
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
CTDSP1 Q9GZU7 1/20 0.38
PTGS2 P35354 1/20 0.37
POLB P06746 1/20 0.37
PDE5A O76074 1/20 0.37
PDE1A P54750 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11233960 0.82 ALDH1A1 (0.44) GAATRPA1MEN1KMT2ANR4A1
SCHEMBL9548043 0.77 RARB (0.47) NPC1RAB9ACYP1A2CYP3A4CYP2C19
SCHEMBL11234022 0.74 CA1 (0.40) GAACLCN2MRGPRX4MEN1KMT2A
Chlorobenzene SCHEMBL17841044 0.72 FOLH1 (0.52) GAACLCN2MRGPRX4NR4A1NPC1
SCHEMBL27890108 0.72 MYC (0.51) GAATRPA1MEN1KMT2ARAB9A
SCHEMBL28854108 0.71 NR4A1 (0.58) GAACLCN2MRGPRX4NR4A1NPC1
SCHEMBL6935726 0.70 TSHR (0.59) CLCN2MRGPRX4SMN1; SMN2
SCHEMBL5113652 0.70 GABRA1 (0.68) CLCN2MRGPRX4
SCHEMBL1457079 0.69 GABRA1 (0.69) CLCN2MRGPRX4
SCHEMBL11390813 0.69 GAA (0.48) GAAMEN1KMT2ARAB9ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4362892-A ARALKYLANILINES, ANTICHOLESTEROL AGENTS BEECHAM GROUP LIMITED (GB) 1982-12-07 US disclosed
US-4206145-A ALKANOYL-SUBSTITUTED ARALKYLAMINES BEECHAM GROUP LIMITED (GB) 1980-06-03 US disclosed