SCHEMBL11234674

SCHEMBL11234674

C=CCc1ccc(-c2ccccc2C(N)=O)nn1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCAT2 O15382 1/20 0.45
KDM4E B2RXH2 2/20 0.40
CSNK1A1 P48729 1/20 0.38
TYRO3 Q06418 1/20 0.38
DYRK1B Q9Y463 1/20 0.38
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
GRM5 P41594 1/20 0.35
KEAP1 Q14145 1/20 0.35
NFE2L2 Q16236 1/20 0.35
CASP1 P29466 1/20 0.35
PARP1 P09874 3/20 0.35
ALDH1A1 P00352 2/20 0.34
TSHR P16473 2/20 0.34
HSD17B10 Q99714 2/20 0.34
MAPT P10636 1/20 0.34
HPGD P15428 1/20 0.34
NUDT1 P36639 1/20 0.34
CYP3A4 P08684 1/20 0.33
CHEK1 O14757 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28177874 0.74 BCAT2 (0.41) BCAT2KDM4ECSNK1A1TYRO3DYRK1B
SCHEMBL8734298 0.74 BCAT2 (0.59) BCAT2KDM4ENPC1RAB9AKEAP1
SCHEMBL9789603 0.73 BCAT2 (0.49) BCAT2KDM4ECSNK1A1TYRO3DYRK1B
SCHEMBL83923 0.69 KDM4E (0.50) BCAT2KDM4EPARP1ALDH1A1TSHR
SCHEMBL31227244 0.68 BCAT2 (0.55) BCAT2KDM4ECSNK1A1TYRO3DYRK1B
SCHEMBL1648463 0.68 BCAT2 (0.55) BCAT2KDM4ECSNK1A1TYRO3DYRK1B
SCHEMBL11794524 0.68 GRM5 (0.47) BCAT2KDM4ECSNK1A1TYRO3DYRK1B
Ammonia Solution, Strong SCHEMBL4442413 0.67 KDM4E (0.49) BCAT2KDM4EPARP1ALDH1A1TSHR
SCHEMBL3205428 0.67 PARP1 (0.36) KDM4EPARP1MAPT
SCHEMBL31531876 0.67 BCAT2 (0.53) BCAT2KDM4ECSNK1A1TYRO3DYRK1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4398044-A Synthesis of acetyl-T-alkanes ELI LILLY AND COMPANY (US) 1983-08-09 US disclosed