SCHEMBL11236268

SCHEMBL11236268

CCCC1(CCC)COC(CCn2ccnc2)(Cc2ccc(Cl)cc2Cl)OC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.40
HMOX1 P09601 2/20 0.40
CYP2C9 P11712 3/20 0.39
LMNA P02545 3/20 0.39
GRM6 O15303 1/20 0.39
NR1I2 O75469 1/20 0.39
EGFR P00533 1/20 0.39
NR3C1 P04150 1/20 0.39
ERBB2 P04626 1/20 0.39
CYP17A1 P05093 1/20 0.39
CYP1A2 P05177 1/20 0.39
FYN P06241 1/20 0.39
PGR P06401 1/20 0.39
CHRM2 P08172 1/20 0.39
CHRM4 P08173 1/20 0.39
ABCB1 P08183 1/20 0.39
ADRB1 P08588 1/20 0.39
CYP3A4 P08684 1/20 0.39
ADRA2A P08913 1/20 0.39
ADORA3 P0DMS8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11239858 0.93 HMOX1 (0.40) KCNH2HMOX1CYP2C9LMNAGRM6
SCHEMBL11252422 0.89 HMOX1 (0.41) KCNH2HMOX1CYP2C9LMNAGRM6
SCHEMBL11245098 0.86 CYP2C9 (0.44) KCNH2HMOX1CYP2C9LMNAGRM6
SCHEMBL11244932 0.86 HMOX1 (0.48) HMOX1
SCHEMBL11239102 0.85 HMOX1 (0.47) HMOX1CYP19A1
SCHEMBL11241392 0.84 CYP2C9 (0.43) KCNH2HMOX1CYP2C9LMNAGRM6
SCHEMBL11235289 0.83 POLB (0.40) CYP2C9CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL11246480 0.80 HMOX1 (0.61) HMOX1LMNAUSP2ALDH1A1ALOX15
SCHEMBL11235305 0.79 CYP19A1 (0.42) HMOX1CYP2C9CYP1A2CYP3A4CYP2D6
SCHEMBL11242344 0.79 HMOX1 (0.49) HMOX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0049565-A2 Derivatives of substituted N-alkylimidazoles, their preparation and pharmaceutical compositions containing them SYNTEX (U.S.A.) INC. (US) 1982-04-14 EP disclosed
US-4321272-A Derivatives of substituted N-alkylimidazoles SYNTEX (U.S.A.) INC. (US) 1982-03-23 US disclosed