SCHEMBL11236328

SCHEMBL11236328

COC(=O)C1=C(C)NC2=C(C(=O)CN(Cc3ccccc3)C2)C1c1ccccc1F

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 11/20 0.47
ALDH1A1 P00352 10/20 0.47
HPGD P15428 9/20 0.47
NPSR1 Q6W5P4 3/20 0.47
HSD17B10 Q99714 7/20 0.45
GAA P10253 7/20 0.45
CASP1 P29466 4/20 0.45
CASP7 P55210 4/20 0.45
SMN1; SMN2 Q16637 3/20 0.44
GALR3 O60755 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
ALOX12 P18054 1/20 0.43
CYP2C19 P33261 1/20 0.43
AURKA O14965 1/20 0.41
AURKB Q96GD4 1/20 0.41
LMNA P02545 2/20 0.41
TSHR P16473 2/20 0.41
GLA P06280 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL10977751 0.99 ALDH1A1 (0.46) KDM4EALDH1A1HPGDNPSR1HSD17B10
SCHEMBL10976629 0.91 ALDH1A1 (0.48) KDM4EALDH1A1HPGDNPSR1HSD17B10
SCHEMBL10972608 0.90 HSD17B10 (0.45) KDM4EALDH1A1HPGDNPSR1HSD17B10
Hydrochloric Acid SCHEMBL10977470 0.89 HSD17B10 (0.44) KDM4EALDH1A1HPGDNPSR1HSD17B10
SCHEMBL10981081 0.88 CACNA1C (0.52) KDM4EALDH1A1HPGDNPSR1GAA
SCHEMBL10979981 0.88 ALDH1A1 (0.48) KDM4EALDH1A1HPGDNPSR1HSD17B10
SCHEMBL10973525 0.85 ALDH1A1 (0.44) KDM4EALDH1A1HPGDNPSR1HSD17B10
Hydrochloric Acid SCHEMBL10975527 0.84 ALDH1A1 (0.44) KDM4EALDH1A1HPGDNPSR1HSD17B10
SCHEMBL5075369 0.84 ABCC9 (0.53) KDM4EALDH1A1HPGDNPSR1LMNA
SCHEMBL10978148 0.81 KMT2A (0.53) KDM4EALDH1A1HPGDNPSR1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4321384-A Antihypertensive agents AMERICAN HOME PRODUCTS CORPORATION (US) 1982-03-23 US disclosed