SCHEMBL11237449

SCHEMBL11237449

COc1ccc(-c2nnc(OC)nc2-c2ccc(OC)cc2)cc1

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.53
KDM4E B2RXH2 3/20 0.53
LMNA P02545 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
TDP1 Q9NUW8 1/20 0.53
L3MBTL1 Q9Y468 1/20 0.53
PTGES O14684 3/20 0.49
KMT2A Q03164 3/20 0.49
MEN1 O00255 2/20 0.49
HPGD P15428 1/20 0.46
GPR84 Q9NQS5 2/20 0.45
MAPT P10636 2/20 0.44
TP53 P04637 1/20 0.44
ADORA1 P30542 2/20 0.44
ADORA2A P29274 1/20 0.44
PTGS1 P23219 1/20 0.44
PTGS2 P35354 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11711628 0.85 ALDH1A1 (0.51) ALDH1A1KDM4ELMNANPSR1TDP1
SCHEMBL11245322 0.84 ALDH1A1 (0.46) ALDH1A1KDM4ELMNANPSR1TDP1
SCHEMBL11231697 0.84 KDM4E (0.39) ALDH1A1KDM4ELMNANPSR1TDP1
SCHEMBL11469872 0.84 CACNA2D1 (0.48) ALDH1A1KDM4ELMNANPSR1PTGES
SCHEMBL11239685 0.84 PTGES (0.50) ALDH1A1KDM4ELMNANPSR1TDP1
SCHEMBL11714188 0.83 ADORA2A (0.47) ALDH1A1KDM4ENPSR1TDP1KMT2A
SCHEMBL11338853 0.83 ADORA1 (0.47) ALDH1A1KDM4ELMNANPSR1L3MBTL1
SCHEMBL11268851 0.82 SMN1; SMN2 (0.53) ALDH1A1KDM4ELMNANPSR1TDP1
SCHEMBL11475908 0.82 RAB9A (0.47) ALDH1A1KDM4EL3MBTL1PTGESKMT2A
SCHEMBL11485833 0.82 PTGES (0.51) ALDH1A1KDM4ELMNANPSR1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4318911-A 5,6-Diaryl-1,2,4-triazines as topical antithrombotic agents ELI LILLY AND COMPANY (US) 1982-03-09 US claimed
US-4021553-A 5,6-Diaryl-1,2,4-triazines as topically-active anti-inflammatory agents ELI LILLY AND COMPANY (US) 1977-05-03 US claimed
US-4318911-A 5,6-Diaryl-1,2,4-triazines as topical antithrombotic agents ELI LILLY AND COMPANY (US) 1982-03-09 US disclosed
US-4190725-A ANTIINFLAMMATORY ELI LILLY AND COMPANY (US) 1980-02-26 US disclosed
US-4021553-A 5,6-Diaryl-1,2,4-triazines as topically-active anti-inflammatory agents ELI LILLY AND COMPANY (US) 1977-05-03 US disclosed