SCHEMBL11238459

SCHEMBL11238459

Cc1[nH]c(=O)c(Cl)cc1-c1cccnc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 1/20 0.48
KMT2A Q03164 1/20 0.47
TYMP P19971 1/20 0.47
PDE3B Q13370 4/20 0.46
PDE3A Q14432 4/20 0.46
AURKB Q96GD4 1/20 0.46
INCENP Q9NQS7 1/20 0.46
NPY5R Q15761 2/20 0.45
PDE4A P27815 2/20 0.44
PDE4B Q07343 2/20 0.44
PDE4C Q08493 2/20 0.44
PDE4D Q08499 2/20 0.44
CYP2A6 P11509 2/20 0.44
KDM4E B2RXH2 2/20 0.43
HPGD P15428 2/20 0.43
ALDH1A1 P00352 1/20 0.43
HSD17B10 Q99714 1/20 0.43
PARP10 Q53GL7 1/20 0.43
PARP11 Q9NR21 1/20 0.43
MAOA P21397 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11229727 0.82 PDE3B (0.68) ALKKMT2APDE3BPDE3AAURKB
SCHEMBL11235886 0.82 PDE3B (0.46) KMT2ATYMPPDE3BPDE3AAURKB
SCHEMBL11235848 0.81 PDE3B (0.67) PDE3BPDE3AAURKBINCENPPDE4A
SCHEMBL2673559 0.81 ALK (0.47) ALKKMT2APDE3BPDE3AAURKB
SCHEMBL11236769 0.80 KDM4E (0.50) ALKKMT2APDE3BPDE3AAURKB
SCHEMBL11243997 0.80 ALK (0.46) ALKKMT2APDE3BPDE3AAURKB
SCHEMBL11078693 0.79 MKNK1 (0.56) ALKKMT2APDE3BPDE3AAURKB
SCHEMBL10911458 0.79 PDE3A (0.71) ALKKMT2APDE3BPDE3AAURKB
SCHEMBL11233155 0.78 CYP11B1 (0.46) ALKKMT2APDE3BPDE3AAURKB
SCHEMBL5270008 0.78 ALK (0.56) ALKKMT2AAURKBNPY5RCYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4365065-A 1-(Pyridinyl)-2-(dimethylamino)ethenyl lower-alkyl ketones STERLING DRUG INC. (US) 1982-12-21 US disclosed
US-4313951-A 3-Substituted-6-(lower-alkyl)-5-(pyridinyl)-2(1H)-pyridinones, their cardiotonic use and intermediates therefor STERLING DRUG INC. (US) 1982-02-02 US disclosed