SCHEMBL11243997

SCHEMBL11243997

CNc1cc(-c2cccnc2)c(C)[nH]c1=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 1/20 0.46
KMT2A Q03164 1/20 0.45
NUDT1 P36639 1/20 0.44
PIK3C3 Q8NEB9 1/20 0.44
PDE3B Q13370 3/20 0.43
PDE3A Q14432 3/20 0.43
AURKB Q96GD4 1/20 0.43
INCENP Q9NQS7 1/20 0.43
PDE4A P27815 2/20 0.42
PDE4B Q07343 2/20 0.42
PDE4C Q08493 2/20 0.42
PDE4D Q08499 2/20 0.42
KDM4E B2RXH2 2/20 0.41
HPGD P15428 2/20 0.41
HTR6 P50406 1/20 0.41
ALDH1A1 P00352 1/20 0.41
HSD17B10 Q99714 1/20 0.41
PARP10 Q53GL7 1/20 0.41
PARP11 Q9NR21 1/20 0.41
CYP2C19 P33261 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11235919 0.82 PDE3B (0.63) PDE3BPDE3AAURKBINCENPPDE4A
SCHEMBL11239104 0.82 NPC1 (0.45) ALKKMT2AAURKBKDM4EHPGD
SCHEMBL11238459 0.80 ALK (0.48) ALKKMT2APIK3C3PDE3BPDE3A
SCHEMBL11229727 0.80 PDE3B (0.68) ALKKMT2APIK3C3PDE3BPDE3A
SCHEMBL2673559 0.79 ALK (0.47) ALKKMT2APIK3C3PDE3BPDE3A
SCHEMBL11236769 0.78 KDM4E (0.50) ALKKMT2APDE3BPDE3AAURKB
SCHEMBL11229029 0.77 ALK (0.43) ALKKMT2ANUDT1PIK3C3PDE3B
SCHEMBL11078693 0.77 MKNK1 (0.56) ALKKMT2APDE3BPDE3AAURKB
SCHEMBL10911458 0.77 PDE3A (0.71) ALKKMT2APIK3C3PDE3BPDE3A
SCHEMBL11233155 0.76 CYP11B1 (0.46) ALKKMT2APDE3BPDE3AAURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4365065-A 1-(Pyridinyl)-2-(dimethylamino)ethenyl lower-alkyl ketones STERLING DRUG INC. (US) 1982-12-21 US disclosed
US-4313951-A 3-Substituted-6-(lower-alkyl)-5-(pyridinyl)-2(1H)-pyridinones, their cardiotonic use and intermediates therefor STERLING DRUG INC. (US) 1982-02-02 US disclosed