SCHEMBL11240927

SCHEMBL11240927

COc1ccc(CCC(=O)CCn2ccnc2)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.58
F2RL1 P55085 1/20 0.55
MEN1 O00255 2/20 0.53
KMT2A Q03164 2/20 0.53
ATM Q13315 1/20 0.53
TSHR P16473 2/20 0.53
ALDH1A1 P00352 2/20 0.53
MAPT P10636 2/20 0.53
TP53 P04637 1/20 0.53
CYP1A2 P05177 1/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2D6 P10635 1/20 0.53
CYP2C9 P11712 1/20 0.53
NFKB1 P19838 1/20 0.53
CYP2C19 P33261 1/20 0.53
MTOR P42345 1/20 0.53
RAB9A P51151 1/20 0.53
HIF1A Q16665 1/20 0.53
GMNN O75496 1/20 0.52
LMNA P02545 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8803260 0.88 CYP19A1 (0.63) CYP19A1F2RL1MEN1KMT2ATSHR
SCHEMBL11240600 0.88 CYP19A1 (0.60) CYP19A1MEN1KMT2AATMTSHR
Hydrochloric Acid SCHEMBL411003 0.87 CYP19A1 (0.62) CYP19A1F2RL1MEN1KMT2AATM
Bromide SCHEMBL11242765 0.87 CYP19A1 (0.62) CYP19A1F2RL1MEN1KMT2ATSHR
SCHEMBL11256565 0.85 TBXAS1 (0.55) TBXAS1
SCHEMBL11253750 0.85 CYP19A1 (0.55) CYP19A1TBXAS1
SCHEMBL11279378 0.83 CYP19A1 (0.65) CYP19A1TBXAS1
SCHEMBL11237835 0.83 TBXAS1 (0.58) CYP19A1TBXAS1
SCHEMBL11240853 0.82 TBXAS1 (0.57) TBXAS1
Hydrochloric Acid SCHEMBL9996061 0.81 TBXAS1 (0.58) TBXAS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4359475-A SPERMICIDES, MICROBIOCIDES OR ANTICONVULSANTS SYNTEX (U.S.A.) INC. (US) 1982-11-16 US disclosed
EP-0049565-A2 Derivatives of substituted N-alkylimidazoles, their preparation and pharmaceutical compositions containing them SYNTEX (U.S.A.) INC. (US) 1982-04-14 EP disclosed
US-4321272-A Derivatives of substituted N-alkylimidazoles SYNTEX (U.S.A.) INC. (US) 1982-03-23 US disclosed