SCHEMBL11240600

SCHEMBL11240600

COc1ccc(CC(=O)CCn2ccnc2)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 3/20 0.60
TBXAS1 P24557 4/20 0.56
MEN1 O00255 1/20 0.54
KMT2A Q03164 1/20 0.54
ATM Q13315 1/20 0.54
ALDH1A1 P00352 3/20 0.54
TSHR P16473 2/20 0.54
MAPT P10636 1/20 0.54
GAA P10253 1/20 0.52
KDM4E B2RXH2 1/20 0.49
TP53 P04637 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2D6 P10635 1/20 0.48
CYP2C9 P11712 1/20 0.48
NFKB1 P19838 1/20 0.48
CYP2C19 P33261 1/20 0.48
MTOR P42345 1/20 0.48
RAB9A P51151 1/20 0.48
HIF1A Q16665 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11238134 0.92 MEN1 (0.59) CYP19A1TBXAS1MEN1KMT2AATM
SCHEMBL11240927 0.88 CYP19A1 (0.58) CYP19A1TBXAS1MEN1KMT2AATM
SCHEMBL11241508 0.86 CYP19A1 (0.66) CYP19A1TBXAS1ALDH1A1TSHRMAPT
SCHEMBL11249784 0.85 TBXAS1 (0.65) CYP19A1TBXAS1ALDH1A1GAAKDM4E
SCHEMBL11236509 0.85 ALDH1A1 (0.55) CYP19A1TBXAS1ALDH1A1MAPTKDM4E
SCHEMBL11259784 0.85 TBXAS1 (0.55) TBXAS1ALDH1A1KDM4EQPCT
SCHEMBL11236348 0.85 CYP19A1 (0.56) CYP19A1TBXAS1ALDH1A1QPCTCYP11B1
SCHEMBL11260419 0.83 TBXAS1 (0.59) TBXAS1
SCHEMBL11242023 0.83 KMT2A (0.53) TBXAS1MEN1KMT2ACYP1A2CYP3A4
SCHEMBL11233236 0.82 HMOX1 (0.57) CYP19A1TBXAS1CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4359475-A SPERMICIDES, MICROBIOCIDES OR ANTICONVULSANTS SYNTEX (U.S.A.) INC. (US) 1982-11-16 US disclosed
EP-0049565-A2 Derivatives of substituted N-alkylimidazoles, their preparation and pharmaceutical compositions containing them SYNTEX (U.S.A.) INC. (US) 1982-04-14 EP disclosed
US-4321272-A Derivatives of substituted N-alkylimidazoles SYNTEX (U.S.A.) INC. (US) 1982-03-23 US disclosed