SCHEMBL11241761

SCHEMBL11241761

Cc1cncc(C)c1-c1ccc(N)c(N)n1

nearest known ligand 0.30

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.30
CYP3A4 P08684 1/20 0.30
TSHR P16473 1/20 0.30
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11241124 0.77 ROCK2 (0.43) CYP3A4TDP1
SCHEMBL11240092 0.75 TSHR (0.39) ALDH1A1CYP3A4TSHRTDP1
SCHEMBL17875696 0.69 BRD4 (0.44) ALDH1A1CYP3A4TSHR
SCHEMBL29745144 0.68 ATR (0.37)
SCHEMBL30873896 0.68 SMN1; SMN2 (0.44) ALDH1A1CYP3A4TDP1
SCHEMBL23123144 0.68 ATR (0.37)
SCHEMBL11238222 0.67 ADORA2A (0.41) ALDH1A1CYP3A4TSHRTDP1
SCHEMBL11226155 0.66 SIRT2 (0.47) ALDH1A1CYP3A4TDP1
SCHEMBL1326003 0.66 ALDH1A1 (0.39) ALDH1A1CYP3A4TSHRTDP1
SCHEMBL11228950 0.65 MAP2K3 (0.58) ALDH1A1CYP3A4TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4317909-A Preparation of 1,3-dihydro-5-(pyridinyl)-2H-imidazo[4,5-b]pyridin-2-ones STERLING DRUG INC. (US) 1982-03-02 US disclosed
US-4294836-A 1,3-Dihydro-6-(pyridinyl)-2H-imidazo[4,5-b]pyridin-2-ones and -imidazo[4,5-b]-pyridine-2-thiones and their cardiotonic use STERLING DRUG INC. (US) 1981-10-13 US disclosed