SCHEMBL11242427

SCHEMBL11242427

COC(=O)c1cc(F)c(-c2nc(Br)c(C(F)(F)F)[nH]2)cc1OC(C)C

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SOS1 Q07889 1/20 0.35
ULK1 O75385 1/20 0.34
DHODH Q02127 5/20 0.33
LMNA P02545 2/20 0.33
NOTUM Q6P988 2/20 0.33
IDH1 O75874 2/20 0.33
RXFP1 Q9HBX9 2/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HTT P42858 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
PTGES O14684 1/20 0.32
ALPL P05186 1/20 0.31
PDE3B Q13370 1/20 0.31
PDE3A Q14432 1/20 0.31
ROCK2 O75116 1/20 0.31
ROCK1 Q13464 1/20 0.31
P2RX3 P56373 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11263574 0.88 DHODH (0.32) DHODHRXFP1
SCHEMBL11251007 0.86 SOS1 (0.40) SOS1LMNANOTUMRXFP1KDM4E
SCHEMBL11248479 0.86 SOS1 (0.36) SOS1LMNANOTUMRXFP1KDM4E
SCHEMBL11253445 0.85 TDP1 (0.37) SOS1LMNANOTUMRXFP1KDM4E
SCHEMBL11246024 0.84 PDE3B (0.33) PDE3BPDE3AP2RX3
SCHEMBL11252299 0.83 XDH (0.33) PDE3BPDE3AP2RX3
SCHEMBL11240936 0.83 SOS1 (0.40) SOS1LMNANOTUMRXFP1KDM4E
SCHEMBL11260601 0.82 SOS1 (0.41) SOS1LMNANOTUMRXFP1KDM4E
SCHEMBL11252931 0.82 TRPA1 (0.36) PDE3BPDE3AP2RX3
SCHEMBL11251640 0.81 SOS1 (0.37) SOS1LMNANOTUMRXFP1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4314844-A FUNGICIDES ROHM AND HAAS COMPANY (US) 1982-02-09 US disclosed