SCHEMBL11242895

SCHEMBL11242895

Cc1cc(-c2cc([N+](=O)[O-])c(=O)[nH]c2C)cc(C)n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIA1 P42261 3/20 0.42
GRIA2 P42262 3/20 0.42
GRIA3 P42263 3/20 0.42
GRIA4 P48058 3/20 0.42
MAPT P10636 3/20 0.42
GRIN2D O15399 2/20 0.42
GRIN3B O60391 2/20 0.42
GRIN1 Q05586 2/20 0.42
GRIN2A Q12879 2/20 0.42
GRIN2B Q13224 2/20 0.42
GRIN2C Q14957 2/20 0.42
GRIN3A Q8TCU5 2/20 0.42
CYP1A2 P05177 2/20 0.42
LMNA P02545 2/20 0.42
HPGD P15428 2/20 0.42
TSHR P16473 2/20 0.42
BLM P54132 2/20 0.42
CYP3A4 P08684 1/20 0.42
GRIK1 P39086 1/20 0.42
GRIK2 Q13002 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11237972 0.81 PDE3B (0.60) LMNAHPGDTSHRBLMKDM4E
SCHEMBL11233155 0.76 CYP11B1 (0.46) MAPTHPGDKDM4EPDE3BPDE3A
SCHEMBL11241138 0.76 GRIA1 (0.42) GRIA1GRIA2GRIA3GRIA4MAPT
SCHEMBL215905 0.73 KDM4E (0.52) GRIA1GRIA2GRIA3GRIA4MAPT
SCHEMBL10910836 0.71 PDE3A (0.67) LMNAHPGDTSHRBLMCYP3A4
SCHEMBL28457504 0.70 KDM4E (0.49) GRIA1GRIA2GRIA3GRIA4MAPT
SCHEMBL11800255 0.70 ALDH1A1 (0.43) GRIA1GRIA2GRIA3GRIA4MAPT
SCHEMBL9332963 0.69 KDM4E (0.47) GRIA1GRIA2GRIA3GRIA4MAPT
SCHEMBL11229699 0.68 PDE3B (0.43) GRIA1GRIA2GRIA3GRIA4MAPT
SCHEMBL9846127 0.68 MAPT (0.47) GRIA1GRIA2GRIA3GRIA4MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4351941-A Pyridinyl-pyridines STERLING DRUG INC. (US) 1982-09-28 US disclosed
US-4331672-A 5-(Pyridinyl)pyridine-2-hydrazines, their preparation and their cardiotonic use STERLING DRUG INC. (US) 1982-05-25 US disclosed