SCHEMBL11229699

SCHEMBL11229699

CCc1[nH]c(=O)c([N+](=O)[O-])cc1-c1ccnc(C)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 3/20 0.43
PDE3A Q14432 3/20 0.43
CCNC P24863 1/20 0.36
CDK8 P49336 1/20 0.36
CDC7 O00311 1/20 0.35
ROCK2 O75116 1/20 0.35
MAP4K4 O95819 1/20 0.35
CDK2 P24941 1/20 0.35
GSK3B P49841 1/20 0.35
CLK4 Q9HAZ1 1/20 0.35
MKNK2 Q9HBH9 1/20 0.35
IRAK4 Q9NWZ3 1/20 0.35
GRIA1 P42261 2/20 0.35
GRIA2 P42262 2/20 0.35
GRIA3 P42263 2/20 0.35
GRIA4 P48058 2/20 0.35
MAPT P10636 2/20 0.35
GRIN2D O15399 1/20 0.35
GRIN3B O60391 1/20 0.35
LMNA P02545 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11235491 0.85 PDE3B (0.59) PDE3BPDE3ACDC7LMNAHPGD
SCHEMBL11236017 0.80 MAPK1 (0.49) PDE3BPDE3ACCNCCDK8CDC7
SCHEMBL11238599 0.80 PDE3B (0.49) PDE3BPDE3ACCNCCDK8CDC7
SCHEMBL11237609 0.78 CYP11B1 (0.43) PDE3BPDE3ACYP3A4HPGDKDM4E
SCHEMBL11243508 0.77 PDE3B (0.43) PDE3BPDE3ACCNCCDK8CDC7
SCHEMBL11241422 0.77 PDE3B (0.43) PDE3BPDE3ACCNCCDK8CDC7
SCHEMBL11223772 0.77 PDE3A (0.73) PDE3BPDE3ALMNACYP3A4HPGD
SCHEMBL11244158 0.76 CCNC (0.49) PDE3BPDE3ACCNCCDK8CDC7
SCHEMBL11231124 0.76 GRIA1 (0.39) CCNCCDK8CDC7ROCK2MAP4K4
SCHEMBL11227650 0.75 PDE3B (0.60) PDE3BPDE3ACDC7GSK3BLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4351941-A Pyridinyl-pyridines STERLING DRUG INC. (US) 1982-09-28 US disclosed
US-4331672-A 5-(Pyridinyl)pyridine-2-hydrazines, their preparation and their cardiotonic use STERLING DRUG INC. (US) 1982-05-25 US disclosed