SCHEMBL11242898

SCHEMBL11242898

Cc1ccccc1OC(N)C(O)CCCN

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 2/20 0.43
CYP1A2 P05177 4/20 0.40
KDM4E B2RXH2 1/20 0.40
SCN4A P35499 2/20 0.39
CYP2D6 P10635 4/20 0.38
SLC6A2 P23975 4/20 0.38
CYP3A4 P08684 3/20 0.38
HTR2A P28223 3/20 0.38
HRH1 P35367 3/20 0.38
SLC6A4 P31645 3/20 0.38
CHRM1 P11229 2/20 0.38
TSHR P16473 2/20 0.38
ADRA2B P18089 2/20 0.38
HTR2C P28335 2/20 0.38
OPRM1 P35372 2/20 0.38
DRD3 P35462 2/20 0.38
OPRK1 P41145 2/20 0.38
HTR2B P41595 2/20 0.38
SLC6A3 Q01959 2/20 0.38
KCNH2 Q12809 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11163903 0.82 HTR2A (0.36) CYP1A2HTR2AHRH1LMNAKMT2A
SCHEMBL11161993 0.78 NOS2 (0.39) CYP2D6SLC6A2HTR2AHRH1SLC6A4
SCHEMBL11172935 0.78 IRAK4 (0.51) KDM4ECYP3A4TSHROPRK1HTR2B
SCHEMBL6693445 0.78 ALOX15 (0.46) ALOX15CYP1A2KDM4ESCN4ACYP2D6
SCHEMBL4071169 0.75 ALOX15 (0.44) ALOX15CYP1A2KDM4ESCN4ACYP2D6
SCHEMBL11242894 0.70 ALOX15 (0.57) ALOX15CYP1A2KDM4ESCN4ACYP2D6
SCHEMBL5960259 0.70 ALOX15 (0.49) ALOX15CYP1A2KDM4ESCN4ACYP2D6
SCHEMBL27684350 0.68 SCN4A (0.48) ALOX15CYP1A2KDM4ESCN4ACYP2D6
SCHEMBL11244735 0.68 TSHR (0.36) ALOX15CYP1A2SCN4ACYP2D6SLC6A2
SCHEMBL10926266 0.68 HTR1B (0.56) ALOX15KDM4ESCN4ACYP2D6TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4318921-A HYPOTENSIVE AGENTS; ADRENERGIC BLOCKING AGENTS IMPERIAL CHEMICAL INDUSTRIES LIMITED (GB) 1982-03-09 US disclosed