SCHEMBL11244220

SCHEMBL11244220

O=Cc1cn(-c2ccccc2)nc1-c1ccc2ccccc2c1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.71
POLB P06746 3/20 0.67
KMT2A Q03164 7/20 0.66
MEN1 O00255 6/20 0.66
NLRP3 Q96P20 1/20 0.66
ALDH1A1 P00352 7/20 0.64
SMN1; SMN2 Q16637 4/20 0.64
LMNA P02545 1/20 0.64
NFKB1 P19838 1/20 0.64
NFKB2 Q00653 1/20 0.64
RELA Q04206 1/20 0.64
KDM4E B2RXH2 5/20 0.56
HPGD P15428 3/20 0.56
ESR1 P03372 1/20 0.54
PTPN2 P17706 2/20 0.53
PTPN1 P18031 2/20 0.53
CDC25B P30305 2/20 0.53
PTPN11 Q06124 2/20 0.53
PTPN6 P29350 1/20 0.53
THRB P10828 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30511902 1.00 PTGS2 (0.71) PTGS2POLBKMT2AMEN1NLRP3
SCHEMBL26121053 0.89 PTGS2 (0.56) PTGS2POLBKMT2AMEN1NLRP3
SCHEMBL11251722 0.86 PTGS2 (0.71) PTGS2POLBKMT2AMEN1NLRP3
SCHEMBL28358360 0.84 PTGS2 (0.94) PTGS2POLBKMT2AMEN1NLRP3
SCHEMBL3447906 0.84 PTGS2 (1.00) PTGS2POLBKMT2AMEN1NLRP3
SCHEMBL28358398 0.83 MEN1 (0.74) PTGS2POLBKMT2AMEN1ALDH1A1
SCHEMBL28361850 0.83 MEN1 (0.74) PTGS2POLBKMT2AMEN1ALDH1A1
SCHEMBL28358299 0.83 MEN1 (0.74) PTGS2POLBKMT2AMEN1ALDH1A1
SCHEMBL28358072 0.83 PTPN2 (0.53) PTGS2POLBKMT2AMEN1NLRP3
SCHEMBL5820153 0.82 POLB (0.73) PTGS2POLBKMT2AMEN1NLRP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110746355-B Phenylpyrazole compound, pharmaceutical composition, and preparation method and application thereof 中国科学院上海有机化学研究所 2023-08-11 CN disclosed
CN-110746355-A Phenylpyrazole compound, pharmaceutical composition, preparation method and application thereof 中国科学院上海有机化学研究所 2020-02-04 CN disclosed
US-4325962-A ANTIINFLAMMATORY AGENTS, ANALGESICS, ANTIDYRETICS BYK-GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1982-04-20 US disclosed