SCHEMBL1124437

SCHEMBL1124437

O=C(O)/C=C/c1cccc(Cl)c1Cl

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.55
CA1 P00915 1/20 0.53
CA2 P00918 1/20 0.53
NFKB1 P19838 1/20 0.53
CA4 P22748 1/20 0.53
PTGER3 P43115 3/20 0.51
PTGER2 P43116 3/20 0.51
PTGER1 P34995 2/20 0.51
MAPT P10636 3/20 0.48
TBXA2R P21731 2/20 0.48
PTGFR P43088 2/20 0.48
PTGIR P43119 2/20 0.48
PTGDR Q13258 2/20 0.48
LMNA P02545 1/20 0.48
ITGB2 P05107 1/20 0.48
ICAM1 P05362 1/20 0.48
ITGAL P20701 1/20 0.48
PTGER4 P35408 1/20 0.48
PLA2G1B P04054 1/20 0.48
ATG4B Q9Y4P1 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1124438 1.00 PTGS2 (0.55) PTGS2CA1CA2NFKB1CA4
SCHEMBL5009953 0.87 PTGS2 (0.48) PTGS2CA1CA2NFKB1CA4
SCHEMBL7004841 0.85 PTGS2 (0.55) PTGS2NFKB1MAPTLMNANPC1
SCHEMBL7004850 0.85 PTGS2 (0.55) PTGS2NFKB1MAPTLMNANPC1
SCHEMBL211297 0.84 HDAC1 (0.65) CA1CA2NFKB1CA4PTGER3
SCHEMBL29393232 0.84 HDAC1 (0.65) CA1CA2NFKB1CA4PTGER3
SCHEMBL12852987 0.84 HDAC1 (0.65) CA1CA2NFKB1CA4PTGER3
SCHEMBL322878 0.84 HDAC1 (0.65) CA1CA2NFKB1CA4PTGER3
SCHEMBL9652685 0.83 PTGS2 (0.54) PTGS2NFKB1MAPTLMNANPC1
SCHEMBL11462614 0.82 HDAC1 (0.62) CA1CA2NFKB1CA4PTGER3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 49 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118930859-A Cinnamic acid modified polyarylene sulfide and preparation method thereof 新凝合科技(成都)有限公司 2024-11-12 CN disclosed
EP-4367105-A1 N-(1,3,4-OXADIAZOL-2-YL)PHENYLCARBOXAMIDES AS HERBICIDES Bayer Aktiengesellschaft (DE) 2024-05-15 EP disclosed
WO-2023280772-A1 N-(1,3,4-OXADIAZOL-2-YL)PHENYLCARBOXAMIDES AS HERBICIDES BAYER AKTIENGESELLSCHAFT (DE) 2023-01-12 WO disclosed
EP-3713417-A1 HERBICIDALLY ACTIVE BICYCLIC BENZAMIDES Bayer Aktiengesellschaft (DE) 2020-09-30 EP disclosed
EP-3638665-A1 HERBICIDALLY ACTIVE 3-PHENYLISOXAZOLINE-5-CARBOXAMIDES OF TETRAHYDRO AND DIHYDROFURAN CARBOXYLIC ACIDS AND ESTERS Bayer Aktiengesellschaft (DE) 2020-04-22 EP disclosed
US-9598412-B2 Spiroindoline compounds for use as anthelminthics INTERVET INC. (US) 2017-03-21 US disclosed
US-20150057302-A1 SPIROINDOLINE COMPOUNDS FOR USE AS ANTHELMINTHICS INTERVET INC. 2015-02-26 US disclosed
US-8809538-B2 Piperidine-containing compounds and use thereof ARRAY BIOPHARMA INC. (US) 2014-08-19 US disclosed
WO-2014090765-A1 USE OF 1-[2-FLUORO-4-METHYL-5-(2,2,2-TRIFLUOROETHYLSULFINYL)PHENYL]-5-AMINO-3-TRIFLUOROMETHYL)-1 H-1,2,4 TFIA ZOLE FOR CONTROLLING NEMATODES IN NEMATODE-RESISTANT CROPS BAYER CROPSCIENCE AG (DE) 2014-06-19 WO disclosed
EP-2531506-B1 Spiroindoline compounds for use as anthelminthics INTERVET INT BV (NL) 2014-05-14 EP disclosed
US-6506940-B1 Converting sertraline stereoisomer into imine form of sertraline; reducing into cis (1S,4S) sertraline and byproduct stereoisomer of sertraline; recovering cis (1S,4S) sertraline from reaction mixture; repeating SUN PHARMACEUTICALS INDUSTRIES LTD. (IN) 2003-01-14 US disclosed
EP-1264820-A1 NOVEL AMIDE COMPOUNDS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-12-11 EP disclosed
WO-2001049638-A2 A PROCESS FOR CONVERTING STEREOISOMERS OF SERTRALINE INTO SERTRALINE SUN PHARMACEUTICAL INDUSTRIES LTD. (IN) 2001-07-12 WO disclosed
US-5863936-A HETEROCYCLIC ENZYME INHIBITORS AS ANTICANCER AGENTS GERON CORPORATION (US) 1999-01-26 US disclosed
US-5677306-A ANTAGONIZING ALPHA-AMINO-3-HYDROXY-5-METHYL-4-ISOXAZOLEPROPIONIC ACID RECEPTOR, USEFUL FOR TREATING ALL ISCHEMIAS RHONE-POULENC RORER S.A. (FR) 1997-10-14 US disclosed
US-5113477-A Core, cladding, heat resistance HITACHI, LTD. (JP) 1992-05-12 US disclosed
EP-0213892-B1 HERBICIDALLY ACTIVE ENOLS ROHM AND HAAS COMPANY (US) 1992-03-25 EP disclosed
US-5017723-A Psychotropic Agents JOUVEINAL S.A. (FR) 1991-05-21 US disclosed
EP-0351856-A2 Thiazolo[5,4-b]azepine compounds Takeda Chemical Industries, Ltd. (JP) 1990-01-24 EP disclosed
EP-0226020-A2 Plastic optical fibers and transparent resin used therefor HITACHI, LTD. (JP) 1987-06-24 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150057302-A1 SPIROINDOLINE COMPOUNDS FOR USE AS ANTHELMINTHICS PKD2, PKD1, PIR PTGS2 156/4885CA1 3866/4885CA2 2006/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.