SCHEMBL11244575

SCHEMBL11244575

CCOC1CCc2ccccc2C1=NO

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
DRD4 P21917 1/20 0.37
KDM4E B2RXH2 5/20 0.36
TSHR P16473 2/20 0.36
ALDH1A1 P00352 2/20 0.36
TDP1 Q9NUW8 2/20 0.36
MAPT P10636 2/20 0.36
HSD17B10 Q99714 1/20 0.36
GRM1 Q13255 1/20 0.36
BLM P54132 1/20 0.36
PMP22 Q01453 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
NFKB1 P19838 1/20 0.36
CYP2C19 P33261 1/20 0.36
RECQL P46063 1/20 0.36
IDO1 P14902 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6181741 0.83 HPGD (0.41) HPGDL3MBTL1KDM4ETSHRALDH1A1
SCHEMBL3370115 0.74 HPGD (0.49) HPGDL3MBTL1SMN1; SMN2KDM4EALDH1A1
SCHEMBL30363500 0.74 HPGD (0.49) HPGDL3MBTL1SMN1; SMN2KDM4EALDH1A1
SCHEMBL3370114 0.74 HPGD (0.49) HPGDL3MBTL1SMN1; SMN2KDM4EALDH1A1
SCHEMBL10041963 0.74 HPGD (0.49) HPGDL3MBTL1SMN1; SMN2KDM4EALDH1A1
SCHEMBL14461584 0.73 IDO1 (0.59) IDO1ACHE
SCHEMBL6328560 0.71 HPGD (0.44) HPGDL3MBTL1SMN1; SMN2KDM4ETSHR
SCHEMBL6328564 0.71 HPGD (0.44) HPGDL3MBTL1SMN1; SMN2KDM4ETSHR
SCHEMBL8736255 0.71 HPGD (0.44) HPGDL3MBTL1SMN1; SMN2KDM4ETSHR
SCHEMBL5263072 0.70 HRH1 (0.39) HPGDL3MBTL1SMN1; SMN2TSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0011747-B1 AMINOPROPANOL DERIVATIVES OF 6-HYDROXY-2,3,4,5-TETRAHYDRO-1H-1-BENZAZEPIN-2-ONES, PROCESS FOR THEIR PREPARATION, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM BASF Aktiengesellschaft (DE) 1982-05-19 EP disclosed