SCHEMBL11244693

SCHEMBL11244693

CCCS(=O)(=O)NC(C)=O.[NaH]

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.31
DHFR P00374 1/20 0.31
TSHR P16473 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
KDM4E B2RXH2 1/20 0.31
MEN1 O00255 1/20 0.31
ALDH1A1 P00352 1/20 0.31
GAA P10253 1/20 0.31
MAPT P10636 1/20 0.31
KMT2A Q03164 1/20 0.31
HSD17B10 Q99714 1/20 0.31
PLK4 O00444 1/20 0.31
AURKA O14965 1/20 0.31
MAPK13 O15264 1/20 0.31
DAPK3 O43293 1/20 0.31
JAK2 O60674 1/20 0.31
PRKCG P05129 1/20 0.31
CDK1 P06493 1/20 0.31
RPS6KB1 P23443 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7987882 0.98 HPGD (0.35) HPGDSMN1; SMN2DHFRTSHRTDP1
SCHEMBL17188793 0.84 ALDH1A1 (0.37) HPGDSMN1; SMN2KDM4EALDH1A1GAA
SCHEMBL13113281 0.82 FAAH (0.41)
SCHEMBL4296201 0.80 FAAH (0.45)
SCHEMBL4666760 0.80 FAAH (0.45)
SCHEMBL13671233 0.80 FAAH (0.45)
SCHEMBL4668386 0.80 FAAH (0.45)
SCHEMBL11979591 0.80 KDM4E (0.35) HPGDSMN1; SMN2DHFRTSHRTDP1
SCHEMBL4719324 0.79
SCHEMBL5154677 0.78 KDM4E (0.35) HPGDSMN1; SMN2TSHRKDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0008802-B1 ERGOLINE DERIVATIVES, THEIR PREPARATION AND THERAPEUTIC COMPOSITION CONTAINING THEM FARMITALIA CARLO ERBA S.p.A. (IT) 1982-07-21 EP disclosed
US-4321381-A Ergot derivatives FARMITALIA CARLO ERBA S.P.A. (IT) 1982-03-23 US disclosed
US-4252941-A HYPOTENSIVE AGENTS, ANTIPROLACTINIC AGENTS FARMITALIA CARLO ERBA S.P.A. (IT) 1981-02-24 US disclosed
EP-0008802-A1 Ergoline derivatives, their preparation and therapeutic composition containing them FARMITALIA CARLO ERBA S.p.A. (IT) 1980-03-19 EP disclosed