SCHEMBL11244696

SCHEMBL11244696

C#CCN(C(N)=NC#N)c1cccc(-c2csc(NC(=N)N)n2)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATP4A P20648 4/20 0.37
ATP4B P51164 4/20 0.37
ABL1 P00519 3/20 0.37
ROCK2 O75116 1/20 0.35
HDAC3 O15379 4/20 0.35
HDAC1 Q13547 4/20 0.35
HDAC2 Q92769 4/20 0.35
HDAC10 Q969S8 4/20 0.35
HDAC8 Q9BY41 3/20 0.35
HDAC6 Q9UBN7 3/20 0.35
HDAC4 P56524 2/20 0.35
HDAC7 Q8WUI4 2/20 0.35
HDAC11 Q96DB2 2/20 0.35
HDAC9 Q9UKV0 2/20 0.35
HDAC5 Q9UQL6 2/20 0.35
MRE11 P49959 2/20 0.35
CSNK2A2 P19784 1/20 0.35
CSNK2B P67870 1/20 0.35
CSNK2A1 P68400 1/20 0.35
CSNK2A3 Q8NEV1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11252869 0.88 ATP4A (0.37) ATP4AATP4BABL1ROCK2HDAC3
SCHEMBL11260913 0.87 ATP4A (0.39) ATP4AATP4BABL1ROCK2HDAC3
SCHEMBL11257651 0.86 GSTO1 (0.39) ATP4AATP4BABL1ROCK2HDAC3
SCHEMBL11254016 0.85 ATP4A (0.41) ATP4AATP4BABL1ROCK2NPC1
SCHEMBL11245308 0.84 ABL1 (0.41) ATP4AATP4BABL1CSNK2A2CSNK2B
SCHEMBL11250101 0.84 POLB (0.42) ATP4AATP4BABL1ROCK2MRE11
SCHEMBL10673686 0.79 ABL1 (0.39) ATP4AATP4BABL1HDAC3HDAC1
SCHEMBL11244719 0.78 ATP4A (0.47) ATP4AATP4BABL1ROCK2CSNK2A2
SCHEMBL11244678 0.77 MAPT (0.42) ATP4AATP4BABL1ROCK2HDAC3
SCHEMBL11244685 0.77 MAPT (0.42) ATP4AATP4BABL1ROCK2HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4315009-A Antisecretory guanidine derivatives and pharmaceutical compositions containing them IMPERIAL CHEMICAL INDUSTRIES LIMITED (GB) 1982-02-09 US claimed
EP-0003640-B1 ANTISECRETORY GUANIDINE DERIVATIVES, PROCESSES FOR THEIR MANUFACTURE AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1982-01-27 EP claimed
EP-0003640-A2 Antisecretory guanidine derivatives, processes for their manufacture and pharmaceutical compositions containing them IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1979-08-22 EP claimed
US-4315009-A Antisecretory guanidine derivatives and pharmaceutical compositions containing them IMPERIAL CHEMICAL INDUSTRIES LIMITED (GB) 1982-02-09 US disclosed
EP-0003640-B1 ANTISECRETORY GUANIDINE DERIVATIVES, PROCESSES FOR THEIR MANUFACTURE AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1982-01-27 EP disclosed
EP-0003640-A2 Antisecretory guanidine derivatives, processes for their manufacture and pharmaceutical compositions containing them IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1979-08-22 EP disclosed